CYR-101

CYR-101 is a dual antagonist of the serotonin (5-HT) receptor subtype 5-HT2A and sigma-2 (sigma2) receptors (Kis = 7.53 and 8.19 nM, respectively).Formal Name: 2-[[1-[2-(4-fluorophenyl)-2-oxoethyl]-4-piperidinyl]methyl]-2,3-dihydro-1H-isoindol-1-one. CAS Number: 359625-79-9. Molecular Formula: C22H23FN2O2. Formula Weight: 366.4. Purity: >95%. Formulation: (Request formulation change), A solid. Solubility: DMF: 10mg/mL, DMF:PBS (pH 7.2) (1:3): 0.25mg/mL, DMSO: 5mg/mL, Ethanol: 3mg/mL. lambdamax: 229, 244 nm. SMILES: O=C1N(CC2CCN(CC(C3=CC=C(F)C=C3)=O)CC2)CC4=CC=CC=C41. InChi Code: InChI=1S/C22H23FN2O2/c23-19-7-5-17(6-8-19)21(26)15-24-11-9-16(10-12-24)13-25-14-18-3-1-2-4-20(18)22(25)27/h1-8,16H,9-15H2. InChi Key: RNRYULFRLCBRQS-UHFFFAOYSA-N.