CTX-1211 (trifluoroacetate salt)

Item number	Size	Manual	SDS	Delivery time	Price
Cay42081-1	1 mg	-	-	6 - 10 business days*	204.00€
Cay42081-5	5 mg	-	-	6 - 10 business days*	958.00€
Cay42081-10	10 mg	-	-	6 - 10 business days*	1,413.00€
Cay42081-25	25 mg	-	-	6 - 10 business days*	2,520.00€

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A peptide agonist of melanocortin receptors, increases cAMP levels in cells expressing MC1R,... more

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Product information "CTX-1211 (trifluoroacetate salt)"

A peptide agonist of melanocortin receptors, increases cAMP levels in cells expressing MC1R, MC3R, or MC4R (EC50s = 6.2, 3.9, and 2.7, nM, respectively), sensitizes male and female mice to liraglutide-induced reductions in food intake and body weight at 1 mg/kg. Formulation: A solid. InChI: InChI=1S/C49H73N19O9S2.C2HF3O2/c1-26-40(71)63-33(16-9-19-58-48(53)54)42(73)65-35(21-28-11-4-3-5-12-28)44(75)64-34(17-10-20-59-49(55)56)43(74)66-36(22-29-23-60-31-14-7-6-13-30(29)31)45(76)67-37(39(50)70)24-78-79-25-38(46(77)61-26)68-41(72)32(62-27(2)69)15-8-18-57-47(51)52,3-2(4,5)1(6)7/h3-7,11-14,23,26,32-38,60H,8-10,15-22,24-25H2,1-2H3,(H2,50,70)(H,61,77)(H,62,69)(H,63,71)(H,64,75)(H,65,73)(H,66,74)(H,67,76)(H,68,72)(H4,51,52,57)(H4,53,54,58)(H4,55,56,59),(H,6,7)/t26-,32+,33+,34+,35-,36+,37+,38+,/m1./s1. InChIKey: QRLRDGUPSFZYLV-CPUQZFJZSA-N. SMILES: O=C(N[C@@H](CSSC[C@@H](C(N[C@@H]1C)=O)NC([C@@H](NC(C)=O)CCCNC(N)=N)=O)C(N)=O)[C@@H](NC([C@@H](NC([C@H](NC([C@@H](NC1=O)CCCNC(N)=N)=O)CC2=CC=CC=C2)=O)CCCNC(N)=N)=O)CC3=CNC4=CC=CC=C34.OC(C(F)(F)F)=O

Keywords:	Acetyl-Arg-cyclo(Cys-D-Ala-Arg-D-Phe-Arg-Trp-Cys)-NH2, N2-acetyl-L-arginyl-L-cysteinyl-D-alanyl-L-arginyl-D-phenylalanyl-L-arginyl-L-tryptophyl-L-cysteinamide, cyclic (2?8)-disulfide, trifluoroacetate salt
Supplier:	Cayman Chemical
Supplier-Nr:	42081