Helianorphin-19

Helianorphin-19
Item number Size Datasheet Manual SDS Delivery time Quantity Price
TGM-T41183-1mg 1 mg

7 - 10 business days*

1,023.00€
 
Description: Helianorphin-19 is a high affinity, potent and selective kappa-opioid receptor (KOR)... more
Product information "Helianorphin-19"
Description: Helianorphin-19 is a high affinity, potent and selective kappa-opioid receptor (KOR) agonist (Ki = 25 nM, EC50= 45 nM). Helianorphin-19 exhibits approximately 200-fold selectivity for KOR over µ and delta-opioid receptors.In vivoHelianorphin-19 shows potent peripheral analgesic efficacy in a mouse model of visceral pain without affecting motor coordination/sedation. References: Muratspahic et al (2021) Design of a stable cyclic peptide analgesic derived from sunflower seeds that targets the kappa-opioid receptor for the treatment of chronic abdominal pain. J.Med.Chem. 64 9042 PMID: 34162205
Supplier: TargetMol
Supplier-Nr: T41183

Properties

Conjugate: No

Database Information

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: +4°C)
Caution
Our products are for laboratory research use only: Not for administration to humans!
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