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EGFR Peptide myristoylated trifluoroacetate salt
Item number: TGM-TP2951-10mg
Description: EGFR peptide (myristoylated) is a synthetic peptide with an amino acid sequence corresponding to the intracellular region of EGFR, capable of inhibiting PKC activity. Smiles:...
| Keywords: | Myr-Arg-Lys-Arg-Thr-Leu-Arg-Arg-Leu-OH , N-myristoyl-RKRTLRRL , EGFR Peptide (myristoylated) (trifluoroacetate salt) ,... |
| MW: | 1422.73 D |
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Sporidesmolide II
Item number: TGM-TP2952-10mg
Description: Sporidesmolide II is a cyclic depsipeptide that was initially isolated from P. chartarum. Target: Others. Smiles: C(C(C)C)[C@@H]1N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](C(C)C)OC(=O)[C@@H](CC(C)C)NC(=O)[C@@]([C@H](CC)C)(NC(=O)[C@H](C(C)C)OC1=O)[H]
| MW: | 652.86 D |
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CP61
Item number: TGM-TP2971-10mg
Description: CP61, a cyclic peptide, functions as a dual inhibitor of CtBP1/CtBP2. It binds to CtBP1 with an affinity of 3 µM and inhibits both heterodimerization and homodimerization of CtBP2 with an IC50 value of 19 µM. CP61 shows promise for cancer research. Target: Others. Smiles:...
| MW: | 1080.26 D |
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Microcin J25
Item number: TGM-TP2972-10mg
Description: Microcin J25 (MccJ25) is a cyclopeptide antibiotic made up of 21 unmodified amino acid residues. It effectively inhibits the DNA-dependent RNA polymerase (RNAP) of Gram-negative bacteria and exhibits antibacterial activity. Smiles:...
| Keywords: | MccJ25 |
| MW: | 2107.32 D |
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PhAc-ALGP-Dox
Item number: TGM-TP2980-10mg
Description: PhAc-ALGP-Dox is a peptide-drug conjugate and a novel antitumor prodrug. It exhibits a range of IC50 values from 311 nM to 34.25 µM against TNBC (E0771), normal mouse epithelium (HC-11), human TNBC (MDA-MB-231 and MDA-MB-468), human colorectal cancer (LS 174T), and normal human epithelium (HME-1) cells....
| MW: | 1003.94 D |
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APP-018
Item number: TGM-TP2982-10mg
Description: APP-018 (D-4F) is an 18 D-amino acid peptide that mimics apolipoprotein A-I (apoA-I). It enhances the anti-inflammatory properties of high-density lipoprotein (HDL) and is applicable in cardiovascular disease research. Target: Apolipoprotein. Smiles:...
| Keywords: | D-4F |
| MW: | 2310.6 D |
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KRL74
Item number: TGM-TP2983-10mg
Description: KRL74 is a cyclic peptide inhibitor that interferes with the interaction between the p6 domain of the HIV Gag protein and the UEV domain of the human TSG101 protein (p6/UEV), with an IC50 of 5.44 µM and a Kd of 11.9 µM. It also inhibits the budding of HIV from host cells, exhibiting an IC50 of 2 µM in...
| MW: | 981.53 D |
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SVS-1 peptide
Item number: TGM-TP2985-10mg
Description: SVS-1 peptide is an anticancer peptide that selectively targets cancer cells through electrostatic interactions, disrupting the cell membrane structure and inducing cell death. Unlike antimicrobial peptides, the activity of SVS-1 peptide occurs before the complete neutralization of membrane charges....
| MW: | 2031.66 D |
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GNQWFI
Item number: TGM-TP2994-10mg
Description: GNQWFI, an anti-Flt1 peptide, functions as a VEGFR1-specific antagonist. It inhibits interactions between VEGFR1 and various ligands, such as VEGFA, VEGFB, and placental growth factor (PIGF), and suppresses VEGF-induced endothelial cell migration and tubulogenesis. GNQWFI holds potential for research in...
| MW: | 763.84 D |
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4-Amino-D-phenylalanine
Item number: TGM-TP2995-10mg
Description: 4-Amino-D-phenylalanine ([D-Phe(4-NH2)]) is a cyclic pentapeptide that inhibits the binding of CXCL12 to CXCR4 in FC131, with an IC50 value of 0.1 µM. Target: CXCR. Smiles: C([C@H](C(O)=O)N)C1=CC=C(N)C=C1
| Keywords: | 4-NH2-d-Phe |
| MW: | 180.2 D |
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Octaarginine
Item number: TGM-TP3000-10mg
Description: Octaarginine is a cell-penetrating peptide (CPP) known for its membrane-translocating activity. CPP's inherent ability to enter cells makes it useful for delivering various membrane-impermeable bioactive agents intracellularly. Additionally, CPP is employed to transport antimicrobial agents into...
| MW: | 1267.5 D |
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Aselacin C
Item number: TGM-TP3006-10mg
Description: Aselacin C is a cyclic peptide that can be isolated from fungi of the Acremonium spp. Target: Others. Smiles: O=C1OC(C)C(NC(=O)C(NC(=O)CCCCCCCC(=O)C=CC=CCCCCC)CCC(=O)N)C(=O)NCCC(=O)NC(C(=O)NC(C(=O)NC1)CO)CC2=CNC=3C=CC=CC32
| MW: | 907.06 D |
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