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JTP10-?-R9 TFA
Item number: TGM-TP2145-100mg
Description: JTP10-?-R9 TFA is a selective inhibitor of the JNK2 peptide (IC50: 89 nM), demonstrating 10-fold higher selectivity for JNK2 over JNK1 and JNK3. Target: JNK. References: Tamer S. Kao, et al. Development of JNK2-selective peptide inhibitors that inhibit breast cancer cell migration. ACS Chem Biol. 2011...
| MW: | 2860.31 D |
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JTP10-?-TATi TFA
Item number: TGM-TP2146-100mg
Description: JTP10-?-TATi TFA is a selective inhibitor of JNK2 peptide (IC50: 92 nM), demonstrating 10-fold selectivity for JNK2 over JNK1 and JNK3. Target: JNK. References: Tamer S. Kao, et al. Development of JNK2-selective peptide inhibitors that inhibit breast cancer cell migration. ACS Chem Biol. 2011 Jun...
| MW: | 2833.28 D |
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LSKL, Inhibitor of Thrombospondin (TSP-1) (TFA)
Item number: TGM-TP2147-100mg
Description: LSKL, Inhibitor of Thrombospondin (TSP-1) TFA, a tetrapeptide derived from latency-associated protein (LAP)-TGFbeta, acts as a competitive antagonist of TGF-beta1. Target: Others. References: Liao F, et al. LSKL peptide alleviates subarachnoid fibrosis and hydrocephalus by inhibiting TSP1-mediated...
| MW: | 572.62 D |
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LXW7 TFA (1313004-77-1 free base)
Item number: TGM-TP2148-100mg
Description: LXW7 TFA, a cyclic peptide containing Arg-Gly-Asp (RGD), is an integrin alphavbeta3 inhibitor with an anti-inflammatory effect. LXW7 has a high binding affinity to alphavbeta3 integrin (IC50: 0.68 µM). It increases the phosphorylation of VEGFR-2 and activation of ERK1/2. Target: Integrin. References:...
| Keywords: | LXW7 TFA |
| MW: | 934.92 D |
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NP213 TFA (942577-31-3 free base)
Item number: TGM-TP2149-100mg
Description: NP213 TFA is a rapidly acting and first-in-class synthetic antimicrobial peptide (AMP) with anti-fungal activity. It targets the fungal cytoplasmic membrane via membrane perturbation and disruption. Target: Others. References: Mercer DK,et al. Improved Methods for Assessing Therapeutic Potential of...
| Keywords: | NP213 TFA |
| MW: | 1207.32 D |
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Nucleoprotein (396-404) (TFA)
Item number: TGM-TP2150-100mg
Description: Nucleoprotein (396-404) TFA, the 396 to 404 fragment of the lymphocytic choriomeningitis virus (LCMV), is the H-2D(b)-restricted immunodominant epitope used as a molecular model of viral antigen. Target: Others. References: Gairin JE, et al. Optimal lymphocytic choriomeningitis virus sequences...
| Keywords: | NP 396 TFA |
| MW: | 1192.2 D |
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pBD-1 TFA (206367-33-1 free base)
Item number: TGM-TP2151L-100mg
Description: pBD-1 TFA is an endogenous and constitutively expressed antimicrobial peptide (AMP) from porcine tissues, has antimicrobial activities and contributes to mucosal and systemic host defenses in pigs. Target: Antibacterial. References: Zhang G, et al. Molecular cloning and tissue expression of porcine...
| Keywords: | pBD-1 TFA |
| MW: | 7180 D |
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RO27-3225 TFA (274682-89-2 free base)
Item number: TGM-TP2154-100mg
Description: RO27-3225 TFA is a potent and selective agonist of melanocortin 4 receptor (MC4R, EC50: 1 nM and 8 nM for MC4R and MC1R) with neuroprotective and anti-inflammatory effects. RO27-3225 TFA shows ~30-fold selectivity for MC4R over MC3R. Target: Others. References: Benoit SC, et al. A novel selective...
| Keywords: | RO27-3225 TFA |
| MW: | 898.93 D |
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TAK-683 TFA (872719-49-8 free base)
Item number: TGM-TP2156-100mg
Description: TAK-683 TFA is a potent full agonist of the KISS1 receptor (KISS1R, IC50: 170 pM) with improved metabolic stability. It shows agonistic activities to KISS1R (EC50s: 0.96 nM and 1.6 nM for human and rat). Target: Others. References: Tanaka A, et al. Evaluation of pharmacokinetics/pharmacodynamics and...
| Keywords: | TAK-683 TFA |
| MW: | 1412.47 D |
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TAT-DEF-Elk-1 TFA (1220751-16-5 free base)
Item number: TGM-TP2157L-100mg
Description: TAT-DEF-Elk-1 TFA is a cell-penetrating peptide Elk-1 inhibitor, mimics and specifically interferes with the DEF domain of Elk-1. TAT-DEF-Elk-1 blocks Elk-1 phosphorylation and prevents Elk-1 nuclear translocation without interfering with ERK nor MSK1 activation. TAT-DEF-Elk-1 is a useful tool to...
| Keywords: | TAT-DEF-Elk-1 TFA, TDE TFA |
| MW: | 3675.09 D |
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Urocortin, rat TFA (171543-83-2 free base)
Item number: TGM-TP2159-100mg
Description: Urocortin, rat TFA is a neuropeptide and a potent endogenous CRFR agonist (Kis: 0.97 nM, 1.5 nM, and 13 nM for mouse CRF2beta, rat CRF2alpha, and human CRF1). Target: Others. References: Perrin MH, et al. Corticotropin releasing factor receptors and their ligand family. Ann N Y Acad Sci. 1999 Oct...
| Keywords: | Urocortin (Rattus norvegicus) (TFA), Rat urocortin TFA, Urocortin, rat TFA |
| MW: | 4821.28 D |
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D-JBD19 TFA (954134-42-0 free base)
Item number: TGM-TP2162L-100mg
Description: D-JBD19 TFA is a non-permeable peptide with neuroprotective effects. Target: Others. References: Cardozo AK, et al. Cell-permeable peptides induce dose- and length-dependent cytotoxic effects. Biochim Biophys Acta. 2007 Sep,1768(9):2222-34.
| Keywords: | D-JBD19 TFA |
| MW: | 2364.58 D |
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