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H-Val-Pro-Pro-OH TFA (58872-39-2 free base)
Item number: TGM-TP1350-10mg
Description: H-Val-Pro-Pro-OH(TFA), a proline peptide derivative from milk, is an ACE inhibitor with IC50 of 9 M. References: Nakamura Y, et al. Purification and characterization of angiotensin I-converting enzyme inhibitors from sour milk. J Dairy Sci. 1995 Apr,78(4):777-83.
| Keywords: | H-Val-Pro-Pro-OH TFA |
| MW: | 425.4 D |
From 43.00€
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[Arg8]-Vasotocin TFA (113-80-4 free base)
Item number: TGM-TP1352-10mg
Description: [Arg8]-Vasotocin (TFA) is a nonmammalian vertebrate neurohypophyseal peptide. References: Ingram CD, et al [Arg8]vasotocin excites neurones in the dorsal vagal complex in vitro: evidence for an action through novel class(es) of CNS receptors. J Neuroendocrinol. 1994 Aug,6(4):415-22.
| Keywords: | [Arg8]-Vasotocin TFA |
| MW: | 1164.24 D |
From 105.00€
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L-JNKI-1
Item number: TGM-TP1353-10mg
Description: L-JNKI-1, a cell-permeable peptide inhibitor specific for JNK, has been shown to effectively inhibit JNK activity in in vivo studies. References: Zhou MS, et al. Role of c-Jun N-terminal kinase in the regulation of vascular tone. J Cardiovasc Pharmacol Ther. 2010 Mar,15(1):78-83.
| MW: | 3822.44 D |
From 139.00€
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ATI-2341 TFA (1337878-62-2 free base)
Item number: TGM-TP1354-10mg
Description: ATI-2341 is an effective functionally selective allosteric agonist for the c-x-c chemokine receptor type 4 (CXCR4), which ACTS as a biased ligand in favor of G G G G G 1 activation instead of G G G G G 13.ATI-2341 activates the inhibitory heterotrimer G protein (Gi) to promote inhibition of cAMP...
| Keywords: | ATI-2341 TFA |
| MW: | 2370.84 D |
From 105.00€
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Arg-Gly-Glu-Ser(TFA)(93674-97-6,free)
Item number: TGM-TP1355-10mg
Description: Arg-gly-glu -Ser(TFA) is a RGD related polypeptide that controls the inhibition of fibrinogen binding to activated platelets by RGDS. References: Moon C, et al. Synthetic RGDS peptide attenuates lipopolysaccharide-induced pulmonary inflammation by inhibiting integrin signaled MAP kinase pathways. Respir...
| Keywords: | Arg-Gly-Glu-Ser(TFA) |
| MW: | 561.47 D |
From 43.00€
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Sarafotoxin S6c
Item number: TGM-TP2120-100ug
Description: Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively). References: Matsuo et al (1997) Effects of sarafotoxin S6c on antidiuresis and NE overflow induced by stimulation of renal nerves in anesthetized dogs. J.Pharmacol.Exp.Ther. 280 905...
| MW: | 2516 D |
885.00€
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Seglitide
Item number: TGM-TP2122-1mg
Description: Peptide agonist for sst2 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: > 1000 (sst1), 0.2 - 1.5 (sst2), 27 - 36 (sst3), > 127 (sst4), and 0.06 - 23 (sst5). References: Hoyer et al (1994) Molecular pharmacology of somatostatin receptors. Naunyn...
| CAS | 81377-02-8 |
| MW: | 808.98 D |
220.00€
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Somatostatin 1-28
Item number: TGM-TP2124-500ug
Description: Somatostatin receptor agonist, derived from the post-translational cleavage of prosomatostatin. References: Panetta et al (1994) Molecular cloning, functional characterization and chromosomal localization of a human somatostatin receptor (somatostatin receptor type 5) with preferential affinity for...
| MW: | 3149 D |
1,355.00€
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R 892
Item number: TGM-TP2126-1mg
Description: Potent and selective bradykinin B1 receptor antagonist (ID50 values are 2.8 and > 600 nM at B1 and B2 receptors respectively). Exhibits no intrinsic agonist activity and is resistant to aminopeptidase and kininase II (ACE) cleavage. Displays hypertensive activity in vivo. References: Gobeil et al (1996)...
| CAS | 229030-05-1 |
| MW: | 1154.37 D |
170.00€
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RI-STAD 2
Item number: TGM-TP2129-10mg
Description: AKAP disruptor. Selectively binds PKA-RI with high affinity (KD values are 6.2 and 12.1 nM for the RIalpha and beta subunits, respectively) and blocks its interaction with AKAP. Inhibits type I PKA-mediated phosphorylation in live cells. Cell permeable. References: Wang et al (2015) PKA-type I selective...
| MW: | 2401.75 D |
1,646.00€
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26RFa
Item number: TGM-TP2132-1mg
Description: Hypothalamic RFamide-related neuropeptide. Acts as a natural ligand of the orphan receptor GPR103. Exhibits orexigenic acitivity in mice upon central administration. References: Kampe et al (2006) Effect of central administration of QRFP(26) peptide on energy balance and characterization of a second...
| CAS | 881640-56-8 |
| MW: | 2818.18 D |
208.00€
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MARCKS Peptide(151-175), Phosphorylated
Item number: TGM-TP1590-100mg
Description: Myristoylated Alanine-Rich C Kinase Substrate peptide (151-175) is a high affinity Protein Kinase C substrate. References: Glaser M, et al. Myristoylated alanine-rich C kinase substrate (MARCKS) produces reversible inhibition of phospholipase C by sequestering phosphatidylinositol 4,5-bisphosphate in...
| MW: | 3320.8 D |
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