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TCMCB07
Item number: TGM-T80540-50mg
Description: TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor 4 (MC4R), with significant implications in the management of cachexia [1]. Target: Melanocortin Receptor
| CAS | 1456699-27-6 |
| MW: | 1230.46 D |
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Z-Leu-Leu-Leu-fluoromethyl ketone
Item number: TGM-T80542-50mg
Description: Z-Leu-Leu-Leu-fluoromethyl ketone (Z-LLL-FMK) acts as a cysteine protease inhibitor and has demonstrated efficacy in blocking SARS infection, while also providing protection to mice when challenged with T. crassiceps [1] [2].
| Keywords: | Z-LLL-FMK |
| CAS | 371167-61-2 |
| MW: | 507.64 D |
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STE-MEK1(13)
Item number: TGM-T80543-50mg
Description: STE-MEK1(13), a cell-permeable ERK1/2 inhibitor with IC50 values ranging from 13 to 30 µM, impedes the phosphorylation of ERK1/2, as demonstrated in studies [1] [2]. Target: ERK
| Keywords: | ERK Activation Inhibitor Peptide, Ste-MPKKKPTPIQLNP-NH2 |
| CAS | 566872-15-9 |
| MW: | 1757.32 D |
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PTPsigma Inhibitor, ISP
Item number: TGM-T80544-50mg
Description: PTPsigma Inhibitor ISP is a compound that binds to recombinant human PTPs, thereby inhibiting PTPsigma signaling. It has the capability to penetrate membranes and counteract the inhibitory effects of chondroitin sulfate proteoglycan (CSPG) on axonal sprouting in spinal cord injury models. Additionally,...
| MW: | 4318.93 D |
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Thioether-cyclized helix B peptide, CHBP
Item number: TGM-T80546-50mg
Description: Thioether-cyclized helix B peptide (CHBP) enhances metabolic stability and exerts renoprotective effects by promoting autophagy through the inhibition of mTOR C1 and activation of mTOR C2 [1]. Target: mTOR
| CAS | 1453840-35-1 |
| MW: | 1416.52 D |
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mSIRK
Item number: TGM-T80548-100mg
Description: mSIRK (G-Protein betagamma Binding Peptide) is a cell-permeable activator of ERK 1/2 with an EC50 of 2.5-5 µM. It disrupts the interaction between the alpha and betagamma subunits, facilitating alpha subunit dissociation without inducing nucleotide exchange [1]. Target: ERK. Smiles:...
| Keywords: | G-Protein betagamma Binding Peptide |
| CAS | 593267-11-9 |
| MW: | 1948.31 D |
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Calmodulin Kinase IINtide, Myristoylated
Item number: TGM-T80549-50mg
Description: Myristoylated Calmodulin Kinase IINtide (Myr-CaMKIINtide) serves as a selective and noncompetitive inhibitor of CaMKII [1]. Target: CaMK
| Keywords: | Myr-CaMKIINtide |
| MW: | 3497.14 D |
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N-myristoyl-RKRTLRRL
Item number: TGM-T80550-50mg
Description: N-myristoyl-RKRTLRRL is a compound that impedes the binding of protein kinase C (PKC) substrates and inhibits calcium (Ca2+)- and phosphatidylserine (PS)-dependent phosphorylation of histones, exhibiting an IC50 of 5 µM. Additionally, it demonstrates an inhibitory effect on histone phosphorylation with...
| CAS | 152246-40-7 |
| MW: | 1308.71 D |
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Calpain inhibitor V
Item number: TGM-T80551-50mg
Description: Calpain Inhibitor V (Mu-Val-HPh-FMK) is a cell-permeable, irreversible calpain inhibitor with demonstrated anti-chlamydial activity [1]. Target: Antibiotic
| Keywords: | Mu-Val-HPh-FMK |
| CAS | 912476-54-1 |
| MW: | 407.48 D |
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MeOSuc-AAPA-CMK
Item number: TGM-T80553-50mg
Description: MeOSuc-AAPA-CMK is a potent inhibitor of human neutrophil elastase (HNE) [1].
| MW: | 490.94 D |
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Myoregulin
Item number: TGM-T80554-50mg
Description: Myoregulin (MLN peptide), a regulin family member, modulates muscle performance through intracellular calcium handling. It directly interacts with the sarcoplasmic reticulum Ca^2+-ATPase (SERCA), impeding Ca^2+ uptake into the sarcoplasmic reticulum [1] [2]. Target: Calcium Channel
| Keywords: | MLN peptide |
| MW: | 5175.17 D |
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wt hMLN
Item number: TGM-T80556-50mg
Description: Wild-type human myoregulin (wt hMLN) is a microprotein that inhibits the sarcoplasmic reticulum Ca2+ pump (SERCA), playing a crucial role in the regulation of calcium homeostasis in skeletal muscle [1]. Target: Calcium Channel
| MW: | 5194.22 D |
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