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beta-Endorphin (1-27) (human)
Item number: TGM-T80515-50mg
Description: beta-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to µ-, delta-, and kappa-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17, and 39.82 nM, respectively. It inhibits analgesia induced by both beta-Endorphin and etorphine [1][2]. Target: Opioid Receptor
| CAS | 76622-84-9 |
| MW: | 3022.47 D |
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human GALP (3-32)
Item number: TGM-T80516-50mg
Description: Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), as evidenced by competitive binding studies. It demonstrates significant potency in modifying the extracellular acidification rate in SH-SY5Y cells...
| Keywords: | Galanin-like peptide (3-32) |
| MW: | 3102.49 D |
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Ala5-Galanin (2-11)
Item number: TGM-T80517-50mg
Description: Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity constant (Ki) of 258 nM [1]. Target: Neuropeptide Y Receptor
| CAS | 859843-84-8 |
| MW: | 1120.3 D |
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Mambalgin-3
Item number: TGM-T80518-50mg
Description: Mambalgin-3, an acid-sensitive ion channel 1 (ASIC1) inhibitor, has potential applications in analgesia research [1]. Target: Sodium Channel
| MW: | 6566.54 D |
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m3-Huwentoxin IV
Item number: TGM-T80519-50mg
Description: m3-Huwentoxin IV (m3-HwTx-IV) is a potent inhibitor of sodium channels (NaV), with half-maximal inhibitory concentrations (IC50s) of 3.3 nM for hNaV1.7, 6.8 nM for hNaV1.6, 7.2 nM for hNaV1.3, 8.4 nM for hNaV1.1, 11.9 nM for hNaV1.2, and 369 nM for hNaV1.4 in the QPatch assay. It also alleviates...
| Keywords: | m3-HwTx-IV |
| MW: | 3985.69 D |
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omega-conotoxin MoVIA
Item number: TGM-T80520-50mg
Description: omega-Conotoxin MVIIA is a potent, selective inhibitor of Ca_v2.2, exhibiting an IC_50 of 0.33 µM in the SH-SY5Y fluorimetric hCa_v2.2 assay [1]. Target: Calcium Channel
| MW: | 3607.15 D |
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Caveolin-1 (82-101) amide (human, mouse, rat)
Item number: TGM-T80521-50mg
Description: Caveolin-1 (82-101) amide (human, mouse, rat), also known as Caveolin-1 scaffolding domain peptide, mitigates aging-related detrimental alterations in various organs and inhibits tyrosine kinases [1]. Target: c-Met/HGFR
| Keywords: | Caveolin-1 scaffolding domain peptide |
| CAS | 2757108-69-1 |
| MW: | 2516.85 D |
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Azurin p28 peptide
Item number: TGM-T80523-50mg
Description: Azurin p28 peptide, a tumor-penetrating antitumor agent, stabilizes p53 by reducing its proteasomal degradation via the formation of a p28:p53 complex. It elicits apoptosis or cell cycle arrest and suppresses the growth of p53-positive tumors. Additionally, the peptide exhibits antiangiogenic properties...
| CAS | 897026-25-4 |
| MW: | 2914.18 D |
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Vm24-toxin
Item number: TGM-T80524-50mg
Description: Vm24-toxin, a peptide toxin isolated from the Mexican scorpion Vaejovis mexicanus smithi, serves as an inhibitor of the Kv1.3 potassium channel [1]. Target: Potassium Channel
| Keywords: | Vaejovis mexicanus peptide 24 |
| CAS | 1373890-79-9 |
| MW: | 3863.59 D |
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E70K
Item number: TGM-T80525-50mg
Description: E70K, a CXCL8 C-terminal peptide, features a lysine (K) substitution for glutamic acid (E) at position 70 and has demonstrated the ability to attenuate neutrophil adhesion and migration in the context of inflammation [1]. Target: CXCR
| MW: | 2400.78 D |
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L-K6L9
Item number: TGM-T80526-50mg
Description: L-K6L9 exhibits antimicrobial and antibiofilm properties effective against P. aeruginosa associated with cystic fibrosis, demonstrating both stability and resistance to degradation by sputum proteases from cystic fibrosis patients, without inducing bacterial resistance [1].
| CAS | 507238-92-8 |
| MW: | 1804.48 D |
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D-K6L9
Item number: TGM-T80527-50mg
Description: D-K6L9 exhibits antimicrobial and antibiofilm properties effective against Pseudomonas aeruginosa isolated from patients with cystic fibrosis. The compound demonstrates stability and resistance to degradation by proteases found in cystic fibrosis sputum and does not promote bacterial resistance [1].
| CAS | 426264-61-1 |
| MW: | 1804.48 D |
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