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Phrixotoxin 2
Item number: TGM-T80054-50mg
Description: Phrixotoxin 2 selectively blocks the KV 4.2 and KV 4.3 channels, demonstrating high specificity in its interaction with these voltage-gated ion channels [1]. Target: Potassium Channel
| CAS | 741738-57-8 |
| MW: | 3921.69 D |
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Pandinotoxin Kalpha
Item number: TGM-T80058-50mg
Description: Pandinotoxin Kalpha, a chemical compound extracted from the emperor scorpion (Pandinus imperator) venom, functions as an inhibitor of the A-type potassium channel [1]. Target: Potassium Channel
| CAS | 185529-64-0 |
| MW: | 4033.71 D |
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Hongotoxin-1
Item number: TGM-T80061-50mg
Description: Hongotoxin-1, a chemical compound isolated from the venom of Centruroides limbatus, functions as a potassium channel inhibitor. It exhibits inhibitory concentrations (IC50) for potassium channel subtypes Kv1.1, Kv1.2, Kv1.3, and Kv1.6 at 31 pM, 170 pM, 86 pM, and 6000 pM, respectively [1]. Target:...
| MW: | 4226.13 D |
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Imperatoxin A
Item number: TGM-T80063-50mg
Description: Imperatoxin A, a peptide toxin sourced from the African scorpion Pandinus imperator, functions as an activator of Ca2+-release channels/ryanodine receptors (RyRs), facilitating increased Ca2+ flow from the sarcoplasmic reticulum into the cell [1]. Target: Calcium Channel
| CAS | 172451-37-5 |
| MW: | 3758.35 D |
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Dendrotoxin-I
Item number: TGM-T80064-50mg
Description: Dendrotoxin-I, a neurotoxin from Dendroaspis snake venom, potently blocks K+ channels, specifically targeting voltage-gated potassium channel subunits KV1.1 and KV1.2 [1] [2] [3]. Target: Potassium Channel
| Keywords: | DTX-I |
| CAS | 107950-33-4 |
| MW: | 7149.24 D |
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Calcicludine
Item number: TGM-T80065-50mg
Description: Calcicludine, a protein toxin derived from the green mamba (Dendroaspis angusticeps) venom, selectively inhibits high-voltage-activated, particularly L-type, calcium channels with an IC50 of 88 nM and plays a role in excitatory synaptic transmission [1] [2]. Target: Calcium Channel
| CAS | 178036-64-1 |
| MW: | 6980.13 D |
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ShK toxin
Item number: TGM-T80066-50mg
Description: ShK toxin, isolated from the Caribbean sea anemone (Stichodactyla helianthus), is an inhibitor of the voltage-dependent potassium channel (Kv1.3 channel). It competes with dendrotoxin I and alpha-dendrotoxin in binding to rat brain synaptosomal membranes and promotes acetylcholine release. Additionally,...
| CAS | 172450-46-3 |
| MW: | 4054.8 D |
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Uroguanylin (human)
Item number: TGM-T80067-50mg
Description: Uroguanylin (human) serves as a natural ligand for the Guanylyl Cyclase C (GCC) receptor in metastatic colorectal cancer tumors and exhibits anti-tumor effects in an animal model of human colon cancer [1] [2]. Target: Guanylate cyclase
| CAS | 154525-25-4 |
| MW: | 1667.86 D |
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Slotoxin
Item number: TGM-T80068-50mg
Description: Slotoxin, a peptide extracted from the venom of the Centruroides noxius Hoffmann scorpion, inhibits high-conductance calcium-activated potassium channels with a dissociation constant (Kd) of 1.5 nM [1]. Target: Potassium Channel
| MW: | 4085.82 D |
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PACAP (6-27) (human, ovine, rat)
Item number: TGM-T80069-50mg
Description: PACAP (6-27) (human, ovine, rat) is an antagonist for the PACAP receptor, inhibiting the catecholamine response of the canine adrenal gland to vasoactive intestinal peptide (VIP), making it a valuable compound for research into cardiovascular and neurological disorders [1].
| Keywords: | Pituitary adenylate cyclase-activating peptide (6-27) |
| CAS | 136134-68-4 |
| MW: | 2638.09 D |
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PKCbetaII Peptide Inhibitor I
Item number: TGM-T80070-50mg
Description: PKCbetaII Peptide Inhibitor I, a specific PKCbetaII inhibitor, exhibits cardioprotective properties in a rat cardiac ischemia/reperfusion injury model and mitigates vascular endothelial dysfunction [1]. Target: PKC
| CAS | 862502-26-9 |
| MW: | 1299.47 D |
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PKCzeta/iota pseudosubstrate inhibitor
Item number: TGM-T80071-1mg
Description: PKCzeta/iota pseudosubstrate inhibitor demonstrates comprehensive inhibitory activity across the protein kinase C (PKC) family and is associated with the induction of memory impairment [1].
| Application: | PKCzeta inhibitor |
| CAS | 799764-07-1 |
| MW: | 1718.02 D |
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