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GR 94800 TFA
Item number: TGM-T75880-50mg
Description: GR 94800 TFA is a potent, selective antagonist of the NK 2 receptor peptide, demonstrating pK B values of 9.6 for NK 2, 6.4 for NK 1, and 6.0 for NK 3 receptors, respectively [1] [2].
| MW: | 1018.08 D |
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GR 64349 TFA
Item number: TGM-T75881-50mg
Description: GR 64349 is a potent and highly selective NK2 receptor peptide antagonist with an EC50 of 3.7 nM in rat colon, exhibiting over 1000-fold selectivity against NK1 receptors and over 300-fold selectivity against NK3 receptors, ensuring targeted action [1] [2].
| MW: | 1035.13 D |
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[Lys5,MeLeu9,Nle10]-NKA(4-10) TFA
Item number: TGM-T75882-50mg
Description: [Lys5,MeLeu9,Nle10]-NKA(4-10) TFA is a potent and highly selective NK2 receptor agonist with an IC50 value of 6.1 nM [1].
| MW: | 918.01 D |
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Agitoxin-2 TFA
Item number: TGM-T75883-50mg
Description: Agitoxin-2 TFA, a potent inhibitor of K+ channels, exhibits IC50 values of 201 pM and 144 pM for mK V 1.3 and mK V 1.1, respectively [1] [2].
| MW: | 4204.89 D |
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PKC beta pseudosubstrate TFA
Item number: TGM-T75885-50mg
Description: PKC beta pseudosubstrate TFA is a selective, cell-permeable inhibitor of PKC [1].
| MW: | 4108.84 D |
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[Ala107]MBP(104-118) TFA
Item number: TGM-T75886-50mg
Description: [Ala107]MBP(104-118) TFA is a noncompetitive peptide inhibitor of protein kinase C (PKC), with IC50 values ranging from 46 to 145 µM.
| MW: | 1607.69 D |
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[Ala113]MBP(104-118) TFA
Item number: TGM-T75887-50mg
Description: [Ala113]MBP(104-118) TFA is a peptide inhibitor that acts noncompetitively against protein kinase C (PKC), with inhibitory concentrations (IC50) ranging from 28 to 62 µM [1].
| MW: | 1607.69 D |
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S961 acetate
Item number: TGM-T76043L-50mg
Description: S961 acetate is a selective and high-affinity antagonist of the insulin receptor (IR), demonstrating IC50 values of 0.048 nM for HIR-A, 0.027 nM for HIR-B, and 630 nM for the human insulin-like growth factor I receptor (HIGF-IR) in SPA assays [1].
| MW: | 4864.18 D |
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Elabela(19-32) TFA
Item number: TGM-T76044-50mg
Description: Elabela(19-32) TFA, an effective fragment of ELABELA (ELA), selectively engages with the apelin receptor (APJ). This compound initiates G alphai1 and beta-arrestin-2 signaling, demonstrating EC50 values of 8.6 nM and 166 nM, respectively. It facilitates receptor internalization, lowers arterial...
| MW: | 1821.05 D |
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Colistin A sulfate hydrate
Item number: TGM-T76045-50mg
Description: Colistin A sulfate hydrate, a key constituent of the polymyxin antibiotic Colistin, effectively combats infections from challenging gram-negative bacteria [1].
| MW: | 1285.55 D |
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BigLEN(rat) TFA
Item number: TGM-T76046-50mg
Description: BigLEN(rat) is a potent GPR171 agonist with an EC50 of 1.6 nM [1].
| MW: | 1860.03 D |
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TAK-683 acetate
Item number: TGM-T76048-50mg
Description: TAK-683 acetate is a nonapeptide metastin analog and a potent full agonist of the KISS1 receptor (KISS1R), exhibiting IC 50 =170 pM and enhanced metabolic stability. This compound shows agonistic activities towards KISS1R, with EC 50 values of 0.96 nM and 1.6 nM for human and rat KISS1R, respectively....
| MW: | 1358.5 D |
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