ZM 241385

ZM 241385
Item number Size Datasheet Manual SDS Delivery time Quantity Price
Cay20447-1 1 mg -

6 - 10 business days*

43.00€
Cay20447-5 5 mg -

6 - 10 business days*

125.00€
Cay20447-10 10 mg -

6 - 10 business days*

175.00€
Cay20447-25 25 mg -

6 - 10 business days*

389.00€
 
ZM 241385 is a potent antagonist of A2A adenosine receptors (pIC50 = 9.52 for displacement of... more
Product information "ZM 241385"
ZM 241385 is a potent antagonist of A2A adenosine receptors (pIC50 = 9.52 for displacement of 5'-N-ethylcarboxamidoadenosine from rat phaeochromocytoma cell membranes). It displays little or no activity at other A adenosine receptors. ZM 241385 is active in vivo. It acts as an inverse agonist at constitutively active mutants of the human A2B adenosine receptor.Formal Name: 4-[2-[[7-amino-2-(2-furanyl)[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]amino]ethyl]-phenol. CAS Number: 139180-30-6. Molecular Formula: C16H15N7O2. Formula Weight: 337.3. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMSO: 100mM, Ethanol: 5 mM. lambdamax: 228, 256 nm. SMILES: OC1=CC=C(CCNC2=NC3=NC(C4=CC=CO4)=NN3C(N)=N2)C=C1. InChi Code: InChI=1S/C16H15N7O2/c17-14-20-15(18-8-7-10-3-5-11(24)6-4-10)21-16-19-13(22-23(14)16)12-2-1-9-25-12/h1-6,9,24H,7-8H2,(H3,17,18,19,20,21,22). InChi Key: PWTBZOIUWZOPFT-UHFFFAOYSA-N.
Keywords: 4-[2-[[7-amino-2-(2-furanyl)[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]amino]ethyl]-phenol
Supplier: Cayman Chemical
Supplier-Nr: 20447

Properties

Application: Potent, selective A2A adenosine receptor antagonist
MW: 337.3 D
Formula: C16H15N7O2
Purity: >98%
Format: Crystalline Solid

Database Information

CAS : 139180-30-6| Matching products
KEGG ID : K04266 | Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: -20°C)
Signal Word: Danger
GHS Hazard Pictograms:
H Phrases: H301
P Phrases: P264, P270, P321, P330, P301+P310, P405, P501
Caution
Our products are for laboratory research use only: Not for administration to humans!
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