VT103
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
A TEAD1 inhibitor (IC50 = 1.02 nM), inhibits TEAD autopalmitoylation in HEK293 cells expressing... more
Product information "VT103"
A TEAD1 inhibitor (IC50 = 1.02 nM), inhibits TEAD autopalmitoylation in HEK293 cells expressing TEAD1 but not HEK293 cells expressing TEAD2, TEAD3, or TEAD4 at 3 µM, inhibits palmitoylation of endogenous TEAD1 in NCI-H2373 cells, reduces tumor volume in NCI-H2373 and NCI H226 mesothelioma mouse xenograft models. Formulation: A solid. InChI: InChI=1S/C18H17F3N4O2S/c1-22-28(26,27)14-7-8-16(15(9-14)17-10-25(2)11-23-17)24-13-5-3-12(4-6-13)18(19,20)21/h3-11,22,24H,1-2H3. InChIKey: LLCVDQHLYHBAHR-UHFFFAOYSA-N. SMILES: O=S(NC)(C1=CC(C2=CN(C)C=N2)=C(NC3=CC=C(C(F)(F)F)C=C3)C=C1)=O
| Keywords: | N-methyl-3-(1-methyl-1H-imidazol-4-yl)-4-[[4-(trifluoromethyl)phenyl]amino]-benzenesulfonamide |
| Supplier: | Cayman Chemical |
| Supplier-Nr: | 42327 |
Properties
| Application: | TEAD1 inhibitor |
| Immunogen: | 410.41 |
| MW: | 410.41 D |
| Formula: | C18H17F3N4O2S |
| Purity: | >98% |
| Format: | Solid |
Database Information
| CAS : | 2290608-13-6| Matching products |
| KEGG ID : | K09448 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +20°C (International: -20°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302, H315, H319, H335 |
| P Phrases: | P261, P264, P270, P271, P280, P301+310, P302+352, P304+340, P305+351+338, P312, P321, P330, P332+313, P337+313, P362+364, P403+233, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
Information about the product reference will follow.
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