Vorapaxar
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor... more
Product information "Vorapaxar"
Description: Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM). Target: Protease-activated Receptor. Smiles: CCOC(=O)N[C@@H]1CC[C@@H]2[C@H](C[C@@H]3[C@@H]([C@@H](C)OC3=O)[C@H]2\C=C\c2ccc(cn2)-c2cccc(F)c2)C1. References: Tang W, Huang B, Wang J, et al. A label-free screening approach targeted protease-activated receptor 1 based on dynamic mass redistribution in living cells[J]. RSC Advances. 2017, 7(68): 43005-43013.
| Keywords: | MK-5348 , SCH 530348 |
| Supplier: | TargetMol |
| Supplier-Nr: | T7013 |
Properties
| Application: | Targets coagulation factor II (thrombin) receptor (F2R, PAR1) |
| MW: | 492.58 D |
| Formula: | C29H33FN2O4 |
Database Information
| CAS : | 618385-01-6| Matching products |
| KEGG ID : | K03914 | Matching products |
| Protein Atlas Nr. : | GPCR Modulators/A(nta)gonists |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H371, H373, H400, H410 |
| P Phrases: | P260, P264, P270, P273, P314, P391, P308+P311, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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