SR1664

Item number	Size	Delivery time	Price
TGM-T23389-1mg	1 mg	7 - 10 business days*	46.00€
TGM-T23389-2mg	2 mg	7 - 10 business days*	65.00€
TGM-T23389-5mg	5 mg	7 - 10 business days*	106.00€
TGM-T23389-1mL	1 ml	7 - 10 business days*	118.00€
TGM-T23389-10mg	10 mg	7 - 10 business days*	138.00€
TGM-T23389-25mg	25 mg	7 - 10 business days*	303.00€
TGM-T23389-50mg	50 mg	7 - 10 business days*	540.00€
TGM-T23389-100mg	100 mg	7 - 10 business days*	777.00€
TGM-T23389-500mg	500 mg	7 - 10 business days*	1,602.00€

If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk

Description: SR1664 is a potent and selective PPARgamma inhibitor with potential antidiabetic... more

Close menu

Product information "SR1664"

Description: SR1664 is a potent and selective PPARgamma inhibitor with potential antidiabetic activity. SR1664 binds to PPARgamma and potently inhibits Cdk5-mediated PPARgamma phosphorylation (IC50 = 80 nM, Ki = 28.67 nM) without exhibiting PPARgamma agonist activity. Target: PPAR. Smiles: C[C@H](NC(=O)c1ccc2n(Cc3ccc(cc3)-c3ccccc3C(O)=O)c(C)c(C)c2c1)c1ccc(cc1)[N+]([O-])=O. References: Marciano DP, Kuruvilla DS, Boregowda SV, et al. Pharmacological repression of PPARgamma promotes osteogenesis. Nat Commun. 2015,6:7443. Published 2015 Jun 12.

Keywords:	SR 1664
Supplier:	TargetMol
Supplier-Nr:	T23389

Properties

Application:	Blocks phosphorylation of PPARgamma by Cdk5
MW:	547.6 D
Formula:	C33H29N3O5

Database Information

CAS :	1338259-05-4\| Matching products
KEGG ID :	K08530 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

Information about the product reference will follow. more

Close menu

You will get a certificate here

Go back

Read, write and discuss reviews... more

Close menu

Customer review for "SR1664"

Write a review