Pexacerfont

Item number	Size	Delivery time	Price
TGM-T16475-1mg	1 mg	7 - 10 business days*	42.00€
TGM-T16475-5mg	5 mg	7 - 10 business days*	88.00€
TGM-T16475-1mL	1 ml	7 - 10 business days*	98.00€

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Description: Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing... more

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Product information "Pexacerfont"

Description: Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing factor receptor (IC50: 6.1±0.6 nM for the human CRF1 receptor). Target: CRFR. Smiles: CC[C@@H](C)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(OC)nc1C. References: Zhou L, et al. In vitro and in vivo metabolism and pharmacokinetics of BMS-562086, a potent and orally bioavailable corticotropin-releasing factor-1 receptor antagonist. Drug Metab Dispos. 2012 Jun,40(6):1093-103.

Keywords:	BMS-562086
Supplier:	TargetMol
Supplier-Nr:	T16475

Properties

Application:	Targets corticotropin releasing hormone receptor 1 (CRHR1)
MW:	340.42 D
Formula:	C18H24N6O
Format:	32160405

Database Information

CAS :	459856-18-9\| Matching products
KEGG ID :	K04578 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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