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Item number: TGM-T16475-1mg

Description: Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing factor receptor (IC50: 6.1±0.6 nM for the human CRF1 receptor). Target: CRFR. Smiles: CC[C@@H](C)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(OC)nc1C. References: Zhou L, et al. In vitro and in vivo metabolism and pharmacokinetics of...

Keywords:	BMS-562086
Application:	Targets corticotropin releasing hormone receptor 1 (CRHR1)
CAS	459856-18-9
MW:	340.42 D

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Pexacerfont

Item number: Cay33221-1

Pexacerfont is an antagonist of corticotropin-releasing factor receptor 1 (CRF1, IC50 = 6.1 nM for the human receptor). It is selective for CRF1 in IMR-32 cells (mean IC50 = 10.6 nM) over CFR2beta receptors endogenously expressed in pig choroid plexus membranes (IC50 = >1,000 nM) in radioligand binding assays and...

Keywords:	BMS 562086, DPC-A69448,...
Application:	CRF1 antagonist
CAS	459856-18-9
MW:	340.4 D

From 52.00€ *

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