Opiranserin (hydrochloride)

Opiranserin (hydrochloride)
Item number Size Datasheet Manual SDS Delivery time Quantity Price
Cay45056-1 1 mg -

6 - 10 business days*

80.00€
Cay45056-5 5 mg -

6 - 10 business days*

359.00€
Cay45056-10 10 mg -

6 - 10 business days*

597.00€
Cay45056-25 25 mg -

6 - 10 business days*

1,093.00€
 
A non-opioid analgesic, an inhibitor of GlyT2 (IC50 = 0.86 µM), antagonist of 5-HT2A and P2X3... more
Product information "Opiranserin (hydrochloride)"
A non-opioid analgesic, an inhibitor of GlyT2 (IC50 = 0.86 µM), antagonist of 5-HT2A and P2X3 (IC50s = 1.3 and 0.87 µM, respectively), reduces mechanical allodynia in a rat model of neuropathic pain induced by spinal nerve ligation (ED50 = 80 mg/kg). SMILES: COC1=CC(C(NCC2(N(C)C)CCOCC2)=O)=CC(OC)=C1OCCCC.Cl. InChi Code: InChI=1S/C21H34N2O5.ClH/c1-6-7-10-28-19-17(25-4)13-16(14-18(19)26-5)20(24)22-15-21(23(2)3)8-11-27-12-9-21,/h13-14H,6-12,15H2,1-5H3,(H,22,24),1H. InChi Key: GSCGQHXDHYVKOL-UHFFFAOYSA-N
Keywords: VVZ-149, 4-butoxy-N-[[4-(dimethylamino)tetrahydro-2H-pyran-4- yl]methyl]-3,5-dimethoxy-benzamide, monohydrochloride
Supplier: Cayman Chemical
Supplier-Nr: 45056

Properties

Application: Non-opioid analgesic, GlyT2 inhibitor
MW: 430.97 D
Formula: C21H34N2O5 . HCl
Purity: >98%
Format: Solid

Database Information

CAS : 1440796-75-7| Matching products
KEGG ID : K05038 | Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: -20°C)
Caution
Our products are for laboratory research use only: Not for administration to humans!
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