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Opiranserin (hydrochloride)
Item number: Cay45056-1
A non-opioid analgesic, an inhibitor of GlyT2 (IC50 = 0.86 µM), antagonist of 5-HT2A and P2X3 (IC50s = 1.3 and 0.87 µM, respectively), reduces mechanical allodynia in a rat model of neuropathic pain induced by spinal nerve ligation (ED50 = 80 mg/kg). SMILES: COC1=CC(C(NCC2(N(C)C)CCOCC2)=O)=CC(OC)=C1OCCCC.Cl. InChi...
| Keywords: | VVZ-149, 4-butoxy-N-[[4-(dimethylamino)tetrahydro-2H-pyran-4- yl]methyl]-3,5-dimethoxy-benzamide, monohydrochloride |
| Application: | Non-opioid analgesic, GlyT2 inhibitor |
| CAS | 1440796-75-7 |
| MW: | 430.97 D |
From 80.00€
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Opiranserin hydrochloride
Item number: TGM-T9833-100mg
Description: Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 µM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 µM). It is development as an injectable agent for the treatment of...
| CAS | 1440796-75-7 |
| MW: | 430.97 D |
From 91.00€
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