MK-0893

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Item number	Size	Manual	Delivery time	Price
Cay28923-1	1 mg	-	6 - 10 business days*	107.00€
Cay28923-5	5 mg	-	6 - 10 business days*	480.00€
Cay28923-10	10 mg	-	6 - 10 business days*	745.00€
Cay28923-25	25 mg	-	6 - 10 business days*	1,198.00€

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A GCGR antagonist (IC50 = 15.7 nM), selective for GCGR over GIPR, GLP-1R, PAC1, VPAC1, and VPAC2... more

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Product information "MK-0893"

A GCGR antagonist (IC50 = 15.7 nM), selective for GCGR over GIPR, GLP-1R, PAC1, VPAC1, and VPAC2 (IC50s = 1,020, >10,000, 9,200, 11,580, and 12,800 nM, respectively), reduces glucagon-induced increases in blood glucose levels in rhesus monkeys at 1 and 3 mg/kg. SMILES: O=C(NCCC(O)=O)C1=CC=C([C@H](C)N2C(C3=CC=C(C=C(OC)C=C4)C4=C3)=CC(C5=CC(Cl)=CC(Cl)=C5)=N2)C=C1. InChi Code: InChI=1S/C32H27Cl2N3O4/c1-19(20-3-5-21(6-4-20)32(40)35-12-11-31(38)39)37-30(18-29(36-37)25-14-26(33)17-27(34)15-25)24-8-7-23-16-28(41-2)10-9-22(23)13-24/h3-10,13-19H,11-12H2,1-2H3,(H,35,40)(H,38,39)/t19-/m0/s1. InChi Key: DNTVJEMGHBIUMW-IBGZPJMESA-N

Keywords:	N-[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-(6-methoxy-2-naphthalenyl)-1H-pyrazol-1-yl]ethyl]benzoyl]-beta-alanine
Supplier:	Cayman Chemical
Supplier-Nr:	28923

Properties

Application:	GCGR antagonist
MW:	588.48 D
Formula:	C32H27Cl2N3O4
Purity:	>98%
Format:	Solid

Database Information

CAS :	870823-12-4\| Matching products
KEGG ID :	K04583 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: -20°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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