GSK973

Item number	Size	Manual	SDS	Delivery time	Price
Cay42057-5	5 mg	-	-	5 - 10 business days*	244.00€
Cay42057-10	10 mg	-	-	5 - 10 business days*	439.00€
Cay42057-25	25 mg	-	-	5 - 10 business days*	972.00€
Cay42057-50	50 mg	-	-	5 - 10 business days*	1,702.00€

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A BET BD2 inhibitor (IC50s = 31.62, 15.85, 15.85, and 39.81 nM for BRD2, BRD3, BRD4, and BRDTBD2,... more

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Product information "GSK973"

A BET BD2 inhibitor (IC50s = 31.62, 15.85, 15.85, and 39.81 nM for BRD2, BRD3, BRD4, and BRDTBD2, respectively), selective for BD2 in BRD2, BRD3, BRD4, and BRDT over BD1 in the same BRDs (IC50s = >10,000 nM for all). Formulation: A solid. InChI: InChI=1S/C23H23FN2O4/c1-25-23(28)15-8-13(22(27)26-20-16-10-29-11-17(16)20)7-14-19(12-5-3-2-4-6-12)18(9-24)30-21(14)15/h2-8,16-20H,9-11H2,1H3,(H,25,28)(H,26,27)/t16-,17+,18-,19+,20+/m1/s1. InChIKey: WZQLVEPIBAOOGF-RMMWZPCPSA-N. SMILES: O=C(C(C=C1[C@@H]2C3=CC=CC=C3)=CC(C(NC)=O)=C1O[C@@H]2CF)N[C@@H]4[C@]5(COC[C@]54[H])[H]

Keywords:	(2S,3S)-2-(fluoromethyl)-2,3-dihydro-N7-methyl-N5-(1a,5beta,6beta)-3-oxabicyclo[3.1.0]hex-6-yl-3-phenyl-5,7-benzofurandicarboxamide
Supplier:	Cayman Chemical
Supplier-Nr:	42057

Properties

Application:	BET BD2 inhibitor
Immunogen:	410.44
MW:	410.44 D
Formula:	C23H23FN2O4
Purity:	>98%
Format:	Solid

Database Information

CAS :	2138473-38-6\| Matching products
KEGG ID :	K11721 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	-20°C (International: -20°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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