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GSK973
Item number: TGM-T39601-5mg
Description: GSK973 is a highly selective and orally bioavailable inhibitor that targets the second bromodomains (BD2s) of the BET family. It exhibits a pIC 50 of 7.8 and a pK d of 8.7 specifically for BRD4 BD2. Additionally, GSK973 demonstrates a remarkable selectivity of 1600-fold for BRD4 BD2 over BRD4 BD1....
| Keywords: | GSK973 |
| CAS | 2138473-38-6 |
| MW: | 410.445 D |
918.00€
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GSK973
Item number: Cay42057-10
A BET BD2 inhibitor (IC50s = 31.62, 15.85, 15.85, and 39.81 nM for BRD2, BRD3, BRD4, and BRDTBD2, respectively), selective for BD2 in BRD2, BRD3, BRD4, and BRDT over BD1 in the same BRDs (IC50s = >10,000 nM for all). Formulation: A solid. InChI:...
| Keywords: | (2S,3S)-2-(fluoromethyl)-2,3-dihydro-N7-methyl-N5-(1a,5beta,6beta)-3-oxabicyclo[3.1.0]hex-6-yl-3-phenyl-5,7-benzofurandica... |
| Application: | BET BD2 inhibitor |
| CAS | 2138473-38-6 |
| MW: | 410.44 D |
From 244.00€
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