GSK046

Item number	Size	Delivery time	Price
TGM-T8932-1mg	1 mg	7 - 10 business days*	114.00€
TGM-T8932-5mg	5 mg	7 - 10 business days*	245.00€
TGM-T8932-1mL	1 ml	7 - 10 business days*	271.00€
TGM-T8932-10mg	10 mg	7 - 10 business days*	395.00€
TGM-T8932-25mg	25 mg	7 - 10 business days*	660.00€
TGM-T8932-50mg	50 mg	7 - 10 business days*	944.00€
TGM-T8932-100mg	100 mg	7 - 10 business days*	1,281.00€

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Description: GSK046 (iBET-BD2) is a potent, selective, and orally active BD2 bromodomain... more

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Product information "GSK046"

Description: GSK046 (iBET-BD2) is a potent, selective, and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50 values of 264 nM [BRD2 BD2], 98 nM [BRD3 BD2], 49 nM [BRD4 BD2], and 214 nM [BRDT BD2], respectively. It exhibits immunomodulatory activity. Target: Epigenetic Reader Domain. Smiles: C[C@H](Oc1cc(cc(F)c1NC(C)=O)C(=O)N[C@H]1CC[C@H](O)CC1)c1ccccc1. References: Omer G, et, al. Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation. Science. 2020 Apr 24, 368(6489): 387-394.

Keywords:	iBET-BD2
Supplier:	TargetMol
Supplier-Nr:	T8932

Properties

Application:	BD2 bromodomain inhibitor
MW:	414.47 D
Formula:	C23H27FN2O4

Database Information

CAS :	2474876-09-8\| Matching products
KEGG ID :	K11721 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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