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GSK046
Item number: TGM-T8932-100mg
Description: GSK046 (iBET-BD2) is a potent, selective, and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50 values of 264 nM [BRD2 BD2], 98 nM [BRD3 BD2], 49 nM [BRD4 BD2], and 214 nM [BRDT BD2], respectively. It exhibits immunomodulatory activity. Target: Epigenetic Reader Domain. Smiles:...
| Keywords: | iBET-BD2 |
| Application: | BD2 bromodomain inhibitor |
| CAS | 2474876-09-8 |
| MW: | 414.47 D |
From 114.00€
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iBET-BD2
Item number: Cay31766-1
iBET-BD2 is an inhibitor of the bromodomain and extra-terminal domain (BET) family protein bromodomain 2 (BD2). It inhibits BD2 in bromodomain-containing protein 2 (BRD2), BRD3, BRD4, and BRDT (IC50s = 264, 98, 49, and 214 nM, respectively) and is selective for BD2 over BD1 (IC50s = 10.96, 36.31, 70.55, and >50.11...
| Keywords: | GSK046, 4-acetamido-3-fluoro-N-((1r,4S)-4-hydroxycyclohexyl)-5-((S)-1-phenylethoxy)benzamide |
| Application: | BD2 bromodomain inhibitor |
| CAS | 2474876-09-8 |
| MW: | 414.5 D |
From 44.00€
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