Grapiprant
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Grapiprant (AAT-007) is a selective EP4 receptor antagonist. Grapiprant displaces... more
Product information "Grapiprant"
Description: Grapiprant (AAT-007) is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM). Target: Prostaglandin Receptor. Smiles: CCc1nc2c(C)nc(C)cc2n1-c1ccc(CCNC(=O)NS(=O)(=O)c2ccc(C)cc2)cc1. References: Vito VD, et al. Detection and quantification of the selective EP4 receptor antagonist CJ-023423 (grapiprant) in canine plasma by HPLC with spectrofluorimetric detection. J Pharm Biomed Anal. 2016 Jan 25,118:251-8.
| Keywords: | AAT-007, CJ-023423, RQ-00000007 |
| Supplier: | TargetMol |
| Supplier-Nr: | TQ0292 |
Properties
| Application: | Targets prostaglandin E receptor 4 (PTGER4) |
| MW: | 491.61 D |
| Formula: | C26H29N5O3S |
Database Information
| CAS : | 415903-37-6| Matching products |
| KEGG ID : | K04261 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302 |
| P Phrases: | P264, P270, P330, P301+P310, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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