CAN508

Item number	Size	Datasheet	Manual	SDS	Delivery time	Price
TGM-T8796-5mg	5 mg				7 - 10 business days*	30.00€
TGM-T8796-1mL	1 ml				7 - 10 business days*	33.00€
TGM-T8796-10mg	10 mg				7 - 10 business days*	39.00€
TGM-T8796-25mg	25 mg				7 - 10 business days*	83.00€
TGM-T8796-50mg	50 mg				7 - 10 business days*	125.00€
TGM-T8796-100mg	100 mg				7 - 10 business days*	187.00€
TGM-T8796-200mg	200 mg	-	-	-	7 - 10 business days*	274.00€

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Description: CAN508 is a potent ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 µM.... more

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Product information "CAN508"

Description: CAN508 is a potent ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 µM. It also competitively inhibits Cdk2-cyclin E with respect to ATP, with Ki and IC50 values of 13.3 µM and 20 µM, respectively. CAN508 exhibits a 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes. [Antitumor activity.]. Target: CDK. Smiles: Nc1n[nH]c(N)c1\N=N\c1ccc(O)cc1. References: Tong Z, et al. Antitumor effects of cyclin dependent kinase 9 inhibition in esophageal adenocarcinoma. Oncotarget. 2017,8(17):28696-28710.

Supplier:	TargetMol
Supplier-Nr:	T8796

Properties

Application:	CDK9 inhibitor
MW:	218.22 D
Formula:	C9H10N6O

Database Information

CAS :	140651-18-9\| Matching products
KEGG ID :	K02211 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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