BX795
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity... more
Product information "BX795"
Description: BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity is 140- and 1600-fold for PDK1 over PKA and PKC in cell-free assays, respectively. Meanwhile, the selectivity for PDK1 is 100-fold than GSK3beta. Target: IkappaB/IKK, Chk, CDK, Autophagy, c-Kit, PDK. Smiles: Ic1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCCNC(=O)c1cccs1. References: Feldman RI, et al. J Biol Chem. 2005, 280(20), 19867-119874.
| Supplier: | TargetMol |
| Supplier-Nr: | T1830 |
Properties
| Application: | PDKP1 inhibitor |
| MW: | 591.47 D |
| Formula: | C23H26IN7O2S |
Database Information
| CAS : | 702675-74-9| Matching products |
| KEGG ID : | K06276 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302, H315, H319, H335 |
| P Phrases: | P261, P264, P270, P271, P280, P301+310, P302+352, P304+340, P305+351+338, P312, P321, P330, P332+313, P337+313, P362+364, P403+233, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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