BI-671800

Item number	Size	Delivery time	Price
TGM-T14565-1mg	1 mg	7 - 10 business days*	54.00€
TGM-T14565-5mg	5 mg	7 - 10 business days*	133.00€
TGM-T14565-1mL	1 ml	7 - 10 business days*	145.00€
TGM-T14565-10mg	10 mg	7 - 10 business days*	217.00€
TGM-T14565-25mg	25 mg	7 - 10 business days*	390.00€
TGM-T14565-50mg	50 mg	7 - 10 business days*	555.00€
TGM-T14565-100mg	100 mg	7 - 10 business days*	756.00€

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Description: BI-671800 (AP-761) is a highly specific and potent antagonist of chemoattractant... more

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Product information "BI-671800"

Description: BI-671800 (AP-761) is a highly specific and potent antagonist of chemoattractant receptor-homologous molecule on Th2 cells (DP2/CRTH2). With IC50 values of 4.5 nM and 3.7 nM for PGD2 binding to CRTH2 in hCRTH2 and mCRTH2 transfected cells, respectively. BI-671800 has the potential to treat poorly controlled asthma[2]. Target: GPR, Prostaglandin Receptor. Smiles: CN(C)c1nc(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)nc(N(C)C)c1CC(O)=O. References: Boehme SA, et al. A small molecule CRTH2 antagonist inhibits FITC-induced allergic cutaneous inflammation. Int Immunol. 2009 Jan,21(1):81-93.

Keywords:	Cmpd A, AP-761
Supplier:	TargetMol
Supplier-Nr:	T14565

Properties

Application:	Prostaglandin D2 receptor CRTH2/GPR44/CD294 antagonist
MW:	501.5 D
Formula:	C25H26F3N5O3

Database Information

CAS :	1093108-50-9\| Matching products
KEGG ID :	K06715 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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