Avapritinib

Item number	Size	Delivery time	Price
TGM-T5109-1mg	1 mg	7 - 10 business days*	81.00€
TGM-T5109-5mg	5 mg	7 - 10 business days*	195.00€
TGM-T5109-1mL	1 ml	7 - 10 business days*	215.00€
TGM-T5109-10mg	10 mg	7 - 10 business days*	320.00€
TGM-T5109-25mg	25 mg	7 - 10 business days*	544.00€
TGM-T5109-50mg	50 mg	7 - 10 business days*	787.00€
TGM-T5109-100mg	100 mg	7 - 10 business days*	1,080.00€
TGM-T5109-500mg	500 mg	7 - 10 business days*	2,183.00€

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Description: Avapritinib (BLU-285) is a dual inhibitor targeting the mutant KIT receptor (KIT... more

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Product information "Avapritinib"

Description: Avapritinib (BLU-285) is a dual inhibitor targeting the mutant KIT receptor (KIT D816V, IC50: 0.27 nM) and PDGFRalpha (PDGFRalpha D842V, IC50: 0.24 nM). Target: c-Kit, PDGFR. Smiles: Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1ccc(F)cc1. References: Erica Evans, et al. Blu-285, a Potent and Selective Inhibitor for Hematologic Malignancies with KIT Exon 17 Mutations.Blood 2015 126:568.

Keywords:	BLU-285
Supplier:	TargetMol
Supplier-Nr:	T5109

Properties

Application:	Targets proto-oncogene tyrosine-protein kinase Kit [EC:2.7.10.1] (KIT, SCFR, CD117)
MW:	498.56 D
Formula:	C26H27FN10
Format:	32160405

Database Information

CAS :	1703793-34-3\| Matching products
KEGG ID :	K04363 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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