ARV-471
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: ARV-471 (Vepdegestrant) is a orally active Cereblon -based estrogen receptor (ER)... more
Product information "ARV-471"
Description: ARV-471 (Vepdegestrant) is a orally active Cereblon -based estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer. Target: Estrogen Receptor/ERR, PROTACs. Smiles: OC=1C=C2C([C@H]([C@H](CC2)C3=CC=CC=C3)C4=CC=C(C=C4)N5CCC(CN6CCN(CC6)C=7C=C8C(=CC7)C(=O)N(C8)[C@@H]9C(=O)NC(=O)CC9)CC5)=CC1. References: John J. Flanagan, et al. ARV-471, an oral estrogen receptor PROTACTM protein degrader for breast cancer. American Association for Cancer Research.2019. 79 (4): P5-04-18.
| Keywords: | Vepdegestrant |
| Supplier: | TargetMol |
| Supplier-Nr: | T39710 |
Properties
| Application: | Targets estrogen receptor alpha (ESR1, NR3A1) |
| MW: | 723.9 D |
| Formula: | C45H49N5O4 |
Database Information
| CAS : | 2229711-68-4| Matching products |
| KEGG ID : | K08550 | Matching products |
| Protein Atlas Nr. : | Gene Regulation |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302, H315, H319 |
| P Phrases: | P264, P270, P280, P321, P330, P301+P310, P302+P352, P305+P351+P338, P332+P313, P337+P313, P362+P364, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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