Apitolisib

Item number	Size	Delivery time	Price
TGM-T1916-2mg	2 mg	7 - 10 business days*	37.00€
TGM-T1916-5mg	5 mg	7 - 10 business days*	55.00€
TGM-T1916-10mg	10 mg	7 - 10 business days*	83.00€
TGM-T1916-25mg	25 mg	7 - 10 business days*	150.00€
TGM-T1916-50mg	50 mg	7 - 10 business days*	243.00€
TGM-T1916-100mg	100 mg	7 - 10 business days*	399.00€

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Description: Apitolisib (RG 7422), an effective, class I PI3K inhibitor for PI3Kalpha(IC50=5 nM),... more

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Product information "Apitolisib"

Description: Apitolisib (RG 7422), an effective, class I PI3K inhibitor for PI3Kalpha(IC50=5 nM), PI3Kbeta(IC50=27 nM), PI3Kdelta(IC50=7 nM), PI3Kgamma (IC50=14 nM), is used in trials study of solid cancers, breast cancer, prostate cancer, renal cell carcinoma, and endometrial carcinoma, among others. Target: Apoptosis, PI3K, mTOR. Smiles: C[C@H](O)C(=O)N1CCN(Cc2sc3c(nc(nc3c2C)-c2cnc(N)nc2)N2CCOCC2)CC1. References: Sutherlin DP, et al. J Med Chem, 2011, 54(21), 7579-7587.

Keywords:	RG 7422, GNE 390, GDC-0980
Supplier:	TargetMol
Supplier-Nr:	T1916

Properties

Application:	Targets phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha/beta/delta
MW:	498.6 D
Formula:	C23H30N8O3S
Format:	32160405

Database Information

CAS :	1032754-93-0\| Matching products
KEGG ID :	K00922 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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