Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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CDK9-Cyclin T1 PPI-IN-1
Item number: TGM-T82758-50mg
Description: CDK9-Cyclin T1 PPI-IN-1 (Compound B19) is a selective inhibitor of the CDK9-Cyclin T1 protein-protein interaction (PPI), suppressing cell proliferation in TNBC MDA-MB-231 cells with an IC50 of 0.044 µM and inducing apoptosis. This compound diminishes CDK9 transcriptional activity and downregulates...
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CDK2-IN-20
Item number: TGM-T82759-50mg
Description: CDK2-IN-20 (compound 3b), a CDK2 inhibitor, exhibits cytotoxic effects on tumor cells with an IC50 ranging from 5.52-17.09 µM. It arrests the MCF-7 cell cycle at the S phase and induces apoptosis [1]. Target: CDK
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C-di-IMP disodium
Item number: TGM-T82760-50mg
Description: C-di-IMP disodium, a STING agonist, is utilized in tumor research [1]. Target: STING
| Keywords: | Cyclic-di-IMP disodium |
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Cd1a
Item number: TGM-T82764-50mg
Description: Cd1a, a beta-toxin from the African spider Ceratogyrus darlingi, modulates calcium ion channels and inhibits human calcium ion channels (Ca v 2.2)(IC 50 2.6 µM) as well as mouse sodium ion channels (Na v 1.7). This compound has potential applications in creating drugs for the treatment of peripheral...
| Keywords: | beta-Theraphotoxin-cd1a, beta-TRTX-cd1a |
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CB2R agonist 3
Item number: TGM-T82769-50mg
Description: CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37µM, indicative of its significant role in the immune system [1]. Target: Cannabinoid Receptor
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CB2R agonist 2
Item number: TGM-T82770-50mg
Description: CB2R agonist 2 (cis-17-para) is a CB2R agonist [1]. Target: Cannabinoid Receptor
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CB2-H
Item number: TGM-T82771-50mg
Description: CB2-H is a dual-channel fluorescent probe for concurrent detection of HOCl and ONOO-, designed to avoid spectral cross-interference. It enables dual-channel fluorescence imaging to monitor endogenously produced HOCl and ONOO- in living cells and zebrafish, responsive to various stimuli [1].
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CB2 receptor antagonist 2
Item number: TGM-T82772-50mg
Description: Compound 39, also known as CB2 receptor antagonist 2, is a potent CB2 antagonist exhibiting an IC50 of 0.33 µM. It engages in strong interactions with residues L17, W6.48, V6.51, and C7.42 [1]. Target: Others
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Caspase-3 activator 3
Item number: TGM-T82774-50mg
Description: Caspase-3 activator 3 (compound 2h) effectively induces apoptosis in HL-60 and K562 cells by substantially activating caspase-3, demonstrating antileukemic activity with IC50 values of 42.89 µM and 33.61 µM, respectively [1]. Target: Caspase
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Caspase-3 activator 2
Item number: TGM-T82775-50mg
Description: Caspase-3 Activator 2 (Compound 2f) is a caspase 3 activator with cytotoxic effects on HL-60 and K562 cells, exhibiting IC 50 values of 33.52 µM and 76.90 µM, respectively [1]. It facilitates apoptosis, rendering it useful in cancer research. Target: Caspase
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Calpurbatug
Item number: TGM-T82788-1mg
Description: Calpurbatug is an immunoglobulin G1 (IgG1) antibody that exhibits affinity for the anti-bacterial DNA-binding protein DNABII family as well as the anti-human monoclonal TRL1068 gamma1-chain [1].
| CAS | 2635404-72-5 |
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Caloxin 1B1
Item number: TGM-T82789-50mg
Description: Caloxin 1B1, a bioactive peptide, exhibits selective inhibition of PMCA extracellularly by binding preferentially to the extracellular domain 1 of PMCA4 over PMCA1. Identified through a screening process for its high-affinity interaction with PMCA, Caloxin 1B1 is capable of direct application to cells...
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