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GSK6853
Item number: Cay20985-5
GSK6853 is a chemical probe for the bromodomain of BRPF1 that displays a TR-FRET pIC50 value of 8.1 and a BROMOscan pKd value of 9.5. It exhibits >1,600-fold selectivity for BRPF1 over all other bromodomains in a BROMOscan assay and shows cellular target engagement with a pIC50 value of 7.7 in a NanoBRET assay...
| Keywords: | N-[2,3-dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxy-benzamide |
| Application: | Peregrin inhibitor |
| CAS | 1910124-24-1 |
| MW: | 409.5 D |
From 44.00€
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GSK-6853
Item number: BPS-82067
GSK-6853 is a potent and selective BRPF1 inhibitor. GSK-6853 exhibits >1600-fold selectivity for BRPF1 over other bromodomains (pIC50 values by TR-FRET are 8.1, 5.1/4.8 and 4.7/<4.3 for BRPF1, BRPF2/3 and BRD4 BD1/2, respectively). The structural analog of GSK-6853, GSK-9311, serves as a good inactive control (125-...
| Keywords: | GSK6853, GSK 6853, |
| Application: | BRPF1 (Peregrin) bromodomain inhibitor |
| CAS | 1910124-24-1 |
| MW: | 409,5 D |
1,123.00€
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