GSK-6853

GSK-6853
Item number Size Datasheet Manual SDS Delivery time Quantity Price
BPS-82067 50 mg - -

3 - 15 business days*

1,123.00€
 
GSK-6853 is a potent and selective BRPF1 inhibitor. GSK-6853 exhibits >1600-fold selectivity for... more
Product information "GSK-6853"
GSK-6853 is a potent and selective BRPF1 inhibitor. GSK-6853 exhibits >1600-fold selectivity for BRPF1 over other bromodomains (pIC50 values by TR-FRET are 8.1, 5.1/4.8 and 4.7/<4.3 for BRPF1, BRPF2/3 and BRD4 BD1/2, respectively). The structural analog of GSK-6853, GSK-9311, serves as a good inactive control (125- and 185-fold reduced potency in cell-free and cell-based assays, respectively).
Keywords: GSK6853, GSK 6853,
Supplier: BPS Bioscience
Supplier-Nr: 82067

Properties

Application: BRPF1 (Peregrin) bromodomain inhibitor
MW: 409,5 D
Formula: C22H27N5O3

Database Information

CAS : 1910124-24-1| Matching products
KEGG ID : K11348 | Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: +20°C)
Caution
Our products are for laboratory research use only: Not for administration to humans!
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