ZB716

Item number	Size	Datasheet	Manual	SDS	Delivery time	Quantity	Price
Cay42238-500	500 µg		-	-	6 - 10 business days*		112.00€
Cay42238-1	1 mg		-	-	6 - 10 business days*		213.00€

If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk

An ERalpha degrader (IC50 = 4.1 nM), inhibits estradiol-induced ERalpha transcriptional activity... more

Close menu

Product information "ZB716"

An ERalpha degrader (IC50 = 4.1 nM), inhibits estradiol-induced ERalpha transcriptional activity in a reporter assay using T47D cells at 1 or 10 nM, decreases the proliferation of MCF-7 and T47D cells and tamoxifen-resistant MCF-7 and T47D cells (IC50s = 0.0032, 0.0062, 0.069, and 0.037 nM, respectively). Formulation: A solid. InChI: InChI=1S/C32H48BF5O4S/c1-30-17-15-26-25-12-11-24(33(40)41)21-23(25)20-22(29(26)27(30)13-14-28(30)39)10-7-5-3-2-4-6-8-18-43(42)19-9-16-31(34,35)32(36,37)38/h11-12,21-22,26-29,39-41H,2-10,13-20H2,1H3/t22-,26-,27+,28+,29-,30+,43?/m1/s1. InChIKey: FIAYIYKWRBIBQG-GDWZZRAASA-N. SMILES: FC(F)(F)C(F)(F)CCCS(CCCCCCCCC[C@H]1[C@]2([H])[C@@](CC[C@]3([C@@]2([H])CC[C@@H]3O)C)([H])C4=CC=C(B(O)O)C=C4C1)=O

Keywords:	Fulvestrant-3 Boronic Acid, B-[(7a,17beta)-17-hydroxy-7-[9-[(4,4,5,5,5-pentafluoropentyl)sulfinyl]nonyl]estra-1,3,5(10)-trien-3-yl]-boronic acid
Supplier:	Cayman Chemical
Supplier-Nr:	42238

Properties

Application:	ERalpha degrader
Immunogen:	634.59
MW:	634.59 D
Formula:	C32H48BF5O4S
Purity:	>95%
Format:	Solid

Database Information

CAS :	1853279-29-4\| Matching products
KEGG ID :	K08550 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: -20°C)
Signal Word:	Danger
GHS Hazard Pictograms:
H Phrases:	H360, H362, H400, H410
P Phrases:	P201, P202, P260, P263, P264, P270, P273, P280, P308+313, P391, P405, P501