Uprosertib
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Uprosertib (GSK2141795) (GSK2141795) is a selective, ATP-competitive, and orally... more
Product information "Uprosertib"
Description: Uprosertib (GSK2141795) (GSK2141795) is a selective, ATP-competitive, and orally bioavailable Akt inhibitor with IC50 of 180 nM, 328 nM, and 38 nM for Akt 1, 2 and 3, respectively. Phase 2. Target: Akt. Smiles: Cn1ncc(Cl)c1-c1cc(oc1Cl)C(=O)NC(CN)Cc1ccc(F)c(F)c1. References: Pachl F, et al. J Proteome Res. 2013, 12(8), 3792-3800.
| Keywords: | GSK2141795, GSK795 |
| Supplier: | TargetMol |
| Supplier-Nr: | T6849 |
Properties
| Application: | Targets RAC serine/threonine-protein kinase [EC:2.7.11.1] (AKT) |
| MW: | 429.25 D |
| Formula: | C18H16Cl2F2N4O2 |
Database Information
| CAS : | 1047634-65-0| Matching products |
| KEGG ID : | K04456 | Matching products |
| Protein Atlas Nr. : | Ser/Thr Phosphorylation |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Danger |
| GHS Hazard Pictograms: |
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| H Phrases: | H372 |
| P Phrases: | P260, P264, P270, P314, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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