Stiripentol
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Stiripentol (BCX2600) (STP) is an anticonvulsant agent, which can inhibit... more
Product information "Stiripentol"
Description: Stiripentol (BCX2600) (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 µM and IC50 of 1.58/3.29 µM, respectively. Target: P450. Smiles: C(=CC(C(C)(C)C)O)C=1C=C2C(=CC1)OCO2. References: Giraud C, et al. In vitro and in vivo inhibitory effect of stiripentol on clobazam metabolism.Drug Metab Dispos. 2006 Apr,34(4):608-11. Epub 2006 Jan 13.
| Keywords: | Diacomit, BCX2600 |
| Supplier: | TargetMol |
| Supplier-Nr: | T4498 |
Properties
| Application: | Synaptosomal GABA uptake inhibitor, CYP3A4 / CYP1A2 / CYP2C19 inhibitor |
| MW: | 234.29 D |
| Formula: | C14H18O3 |
Database Information
| CAS : | 49763-96-4| Matching products |
| KEGG ID : | K17689 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302 |
| P Phrases: | P264, P270, P301+310, P330, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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