Ralaniten
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An antagonist of the androgen receptor NTD, inhibits androgen receptor NTD transactivation in a... more
Product information "Ralaniten"
An antagonist of the androgen receptor NTD, inhibits androgen receptor NTD transactivation in a reporter assay (IC50 = 7.4 µM), reduces androgen-dependent growth of LNCaP cells from 10-30 µM, decreases tumor volume in an LNCaP CRPC mouse xenograft model at 50 mg/kg. Formulation: A solid. InChI: InChI=1S/C21H27ClO5/c1-21(2,15-3-7-19(8-4-15)26-13-17(24)11-22)16-5-9-20(10-6-16)27-14-18(25)12-23/h3-10,17-18,23-25H,11-14H2,1-2H3/t17-,18-/m1/s1. InChIKey: HDTYUHNZRYZEEB-QZTJIDSGSA-N. SMILES: O[C@@H](COC1=CC=C(C(C)(C)C2=CC=C(OC[C@@H](CCl)O)C=C2)C=C1)CO
| Keywords: | EPI-002, (2R)-3-[4-[1-[4-[(2S)-3-chloro-2-hydroxypropoxy]phenyl]-1-methylethyl]phenoxy]-1,2-propanediol |
| Supplier: | Cayman Chemical |
| Supplier-Nr: | 42391 |
Properties
| Application: | Androgen receptor NTD antagonist |
| Immunogen: | 394.89 |
| MW: | 394.89 D |
| Formula: | C21H27ClO5 |
| Purity: | >95% |
| Format: | Solid |
Database Information
| CAS : | 1203490-23-6| Matching products |
| KEGG ID : | K08557 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +20°C (International: -20°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302, H315, H319, H335 |
| P Phrases: | P261, P264, P270, P271, P280, P301+310, P302+352, P304+340, P305+351+338, P312, P321, P330, P332+313, P337+313, P362+364, P403+233, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
Information about the product reference will follow.
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