MRTX0902

Item number	Size	Delivery time	Price
TGM-T9755-1mg	1 mg	7 - 10 business days*	86.00€
TGM-T9755-5mg	5 mg	7 - 10 business days*	212.00€
TGM-T9755-10mg	10 mg	7 - 10 business days*	311.00€
TGM-T9755-25mg	25 mg	7 - 10 business days*	660.00€
TGM-T9755-50mg	50 mg	7 - 10 business days*	1,060.00€
TGM-T9755-100mg	100 mg	7 - 10 business days*	1,731.00€

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Description: MRTX0902 is an effective and high selective inhibitor of SOS1 with an IC50 of 46 nM... more

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Product information "MRTX0902"

Description: MRTX0902 is an effective and high selective inhibitor of SOS1 with an IC50 of 46 nM and a Ki of 2 nM. Target: Raf. Smiles: C[C@@H](Nc1nnc(C)c2cnc(cc12)N1CCOCC1)c1cccc(C#N)c1C. References: Ketcham JM, et al. Design and Discovery of MRTX0902, a Potent, Selective, Brain-Penetrant, and Orally Bioavailable Inhibitor of the SOS1:KRAS Protein-Protein Interaction. J Med Chem. 2022 Jul 28,65(14):9678-9690.

Keywords:	UNII-CRG69FR93G
Supplier:	TargetMol
Supplier-Nr:	T9755

Properties

Application:	SOS1-K-Ras(G12C) protein-protein interaction inhibitor
MW:	388.47 D
Formula:	C22H24N6O

Database Information

CAS :	2654743-22-1\| Matching products
KEGG ID :	K03099 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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