Laropiprant
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2... more
Product information "Laropiprant"
Description: Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such as and DP/DP1 receptor(Ki = 0.57 nM) and TP Receptor(Ki = 2.95 nM). Target: Prostaglandin Receptor. Smiles: CS(=O)(=O)c1cc(F)cc2c3CC[C@H](CC(O)=O)c3n(Cc3ccc(Cl)cc3)c12. References: Sturino CF, et al. Discovery of a potent and selective prostaglandin D2 receptor antagonist, [(3R)-4-(4-chloro-benzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]-acetic acid (MK-0524). J Med Chem. 2007 Feb 22,50(4):794-806.
| Keywords: | MK-0524 |
| Supplier: | TargetMol |
| Supplier-Nr: | T15712 |
Properties
| Application: | Targets prostaglandin D2 receptor (PTGDR) |
| MW: | 435.9 D |
| Formula: | C21H19ClFNO4S |
Database Information
| CAS : | 571170-77-9| Matching products |
| KEGG ID : | K04332 | Matching products |
| Protein Atlas Nr. : | GPCR Modulators/A(nta)gonists |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302 |
| P Phrases: | P264, P270, P330, P301+P310, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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