K-252c
| Item number | Size | Datasheet | Manual | SDS | Delivery time | Quantity | Price |
|---|---|---|---|---|---|---|---|
| TGM-T15638-5mg | 5 mg |
7 - 10 business days* |
807.00€
|
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| TGM-T15638-10mg | 10 mg |
7 - 10 business days* |
1,402.00€
|
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a... more
Product information "K-252c"
Description: K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor (IC50: 2.45 µM). K-252c also inhibits beta-lactamase, chymotrypsin, and malate dehydrogenase. K-252c causes apoptosis in human chronic myelogenous leukemia cancer cells. Target: PKC. Smiles: O=C1NCc2c1c1c3ccccc3[nH]c1c1[nH]c3ccccc3c21. References: Pereira, E.R., et al. Structure-activity relationships in a series of substituted indolocarbazoles: Topoisomerase I and protein kinase C inhibition and antitumoral and antimicrobial properties J. Med. Chem. 39(22), 4471-4477 (1996).
| Supplier: | TargetMol |
| Supplier-Nr: | T15638 |
Properties
| Application: | Indolocarbazole alkaloid antibiotic, PKC inhibitor |
| MW: | 311.34 D |
| Formula: | C20H13N3O |
Database Information
| CAS : | 85753-43-1| Matching products |
| KEGG ID : | K02677 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +20°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302, H319 |
| P Phrases: | P264, P270, P280, P330, P301+P310, P305+P351+P338, P337+P313, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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