Istradefylline
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR)... more
Product information "Istradefylline"
Description: Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in trials studying the treatment and basic science of Drug Abuse, Sleep Disorder, Hepatic Impairment, Parkinson's Disease, and Restless Legs Syndrome, among others. Target: Adenosine Receptor. Smiles: CN1C2=C(N(CC)C(=O)N(CC)C2=O)N=C1/C=C/C3=CC(OC)=C(OC)C=C3. References: Chen JF, et al. J Neurosci, 2001, 21(10), RC143.
| Keywords: | KW-6002 |
| Supplier: | TargetMol |
| Supplier-Nr: | T6552 |
Properties
| Application: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| MW: | 384.43 D |
| Formula: | C20H24N4O4 |
Database Information
| CAS : | 155270-99-8| Matching products |
| KEGG ID : | K04266 | Matching products |
| Protein Atlas Nr. : | GPCR Modulators/A(nta)gonists |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Danger |
| GHS Hazard Pictograms: |
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| H Phrases: | H301 |
| P Phrases: | P264, P270, P321, P330, P301+P310, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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