Irdabisant hydrochloride

Item number	Size	Delivery time	Price
TGM-T61197-25mg	25 mg	7 - 10 business days*	1,520.00€
TGM-T61197-50mg	50 mg	7 - 10 business days*	1,982.00€
TGM-T61197-100mg	100 mg	7 - 10 business days*	2,503.00€

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Description: Irdabisant hydrochloride (CEP-26401) is a selective, orally active, and blood-brain... more

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Product information "Irdabisant hydrochloride"

Description: Irdabisant hydrochloride (CEP-26401) is a selective, orally active, and blood-brain barrier penetrating histamine H3 receptor (H3R) inverse agonist, demonstrating high affinity with K*i values of 7.2 nM and 2.0 nM for rat and human H3R, respectively. Exhibiting relatively low hERG current inhibitory activity with an IC*50 of 13.8 µM, this compound has shown to enhance cognition and promote wakefulness in rat social recognition models, suggesting potential applications in schizophrenia or cognitive impairment research. Target: Others. Smiles: Cl.C[C@@H]1CCCN1CCCOc1ccc(cc1)-c1ccc(=O)[nH]n1

Supplier:	TargetMol
Supplier-Nr:	T61197

Properties

Application:	Targets histamine receptor H3 (HRH3)
MW:	349.86 D
Formula:	C18H24ClN3O2
Format:	32160405

Database Information

CAS :	1005398-61-7\| Matching products
KEGG ID :	K04151 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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