GSK682753A

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Item number	Size	Manual	Delivery time	Price
Cay45381-5	5 mg	-	6 - 10 business days*	189.00€
Cay45381-10	10 mg	-	6 - 10 business days*	301.00€
Cay45381-25	25 mg	-	6 - 10 business days*	657.00€

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An EBI2 inverse agonist, inhibits CREB activity in a reporter assay using HEK293 cells... more

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Product information "GSK682753A"

An EBI2 inverse agonist, inhibits CREB activity in a reporter assay using HEK293 cells transiently transfected with EBI2 and Gqi4myr (IC50 = 53.6 nM), inhibits antibody-induced proliferation of B cells isolated from transgenic mice overexpressing human EBI2 from 0.001-1 µM. SMILES: O=C1OC2(CCN(CC2)C(/C=C/C3=CC=C(C=C3)Cl)=O)CN1CC4=CC(Cl)=C(C=C4)Cl. InChi Code: InChI=1S/C23H21Cl3N2O3/c24-18-5-1-16(2-6-18)4-8-21(29)27-11-9-23(10-12-27)15-28(22(30)31-23)14-17-3-7-19(25)20(26)13-17/h1-8,13H,9-12,14-15H2/b8-4+. InChi Key: RDDLWMWIRXGSJM-XBXARRHUSA-N

Keywords:	8-[(2E)-3-(4-chlorophenyl)-1-oxo-2-propen-1-yl]-3-[(34-,dichlorophenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
Supplier:	Cayman Chemical
Supplier-Nr:	45381

Properties

Application:	EBI2 (GPR183) inverse agonist
MW:	479.78 D
Formula:	C23H21Cl3N2O3
Purity:	>98%
Format:	Solid

Database Information

CAS :	1334294-76-6\| Matching products
KEGG ID :	K04305 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	-20°C (International: -20°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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