GSK2250665A

NEW

Item number	Size	Datasheet	Manual	SDS	Delivery time	Quantity	Price
Cay45942-1	1 mg		-		5 - 10 business days*		91.00€
Cay45942-5	5 mg		-		5 - 10 business days*		408.00€

If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk

GSK2250665A is an IL-2-inducible T cell kinase (Itk) inhibitor (IC50 = 0.63 nM). It is selective... more

Close menu

Product information "GSK2250665A"

GSK2250665A is an IL-2-inducible T cell kinase (Itk) inhibitor (IC50 = 0.63 nM). It is selective for Itk over Aurora B kinase (IC50 = 398 nM) and a panel of 11 kinases (IC50s = 4-631 nM). GSK2250665A reduces the levels of IFN-gamma in isolated human peripheral blood mononuclear cells (PBMCs, IC50 = 25 nM).. SMILES: O[C@@H](CC1)CC[C@H]1NC2=NC(CC3=CC=CC=C3)=CC(NC4=NC5=CC=C(CC)C=C5S4)=N2. InChi Code: InChI=1S/C26H29N5OS/c1-2-17-8-13-22-23(15-17)33-26(29-22)31-24-16-20(14-18-6-4-3-5-7-18)28-25(30-24)27-19-9-11-21(32)12-10-19/h3-8,13,15-16,19,21,32H,2,9-12,14H2,1H3,(H2,27,28,29,30,31)/t19-,21-. InChi Key: DPRNXTSMYVCYLJ-XUTJKUGGSA-N

Keywords:	trans-4-[[4-[(6-ethyl-2-benzothiazolyl)amino]-6-(phenylmethyl)-2-pyrimidinyl]amino]-cyclohexanol
Supplier:	Cayman Chemical
Supplier-Nr:	45942

Properties

Application:	ITK inhibitor
MW:	459.61 D
Formula:	C26H29N5OS
Purity:	>98%
Format:	Solid

Database Information

CAS :	1246030-96-5\| Matching products
KEGG ID :	K07363 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: -20°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

Information about the product reference will follow. more

Close menu

View product citations for antibody 45942 on CiteAb

You will get a certificate here

Go back

Read, write and discuss reviews... more

Close menu

Customer review for "GSK2250665A"

Write a review