GSK-4716
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: GSK4716 is an ERRbeta/gamma agonist (IC50 = 2 µM) that can activate the receptor... more
Product information "GSK-4716"
Description: GSK4716 is an ERRbeta/gamma agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand. Target: Estrogen Receptor/ERR. Smiles: CC(C)c1ccc(\C=N\NC(=O)c2ccc(O)cc2)cc1. References: Wang L , Zuercher W J , Consler T G , et al. X-ray Crystal Structures of the Estrogen-related Receptor-? Ligand Binding Domain in Three Functional States Reveal the Molecular Basis of Small Molecule Regulation[J]. Journal of Biological Chemistry, 2006, 281(49):37773-37781.
| Supplier: | TargetMol |
| Supplier-Nr: | T5531 |
Properties
| Application: | ERR beta/gamma agonist |
| MW: | 282.34 D |
| Formula: | C17H18N2O2 |
Database Information
| CAS : | 101574-65-6| Matching products |
| KEGG ID : | K08552 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H317, H410 |
| P Phrases: | P261, P272, P273, P280, P321, P391, P302+P352, P333+P313, P362+P364, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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