ESI-08

Item number	Size	Delivery time	Price
TGM-T11234-1mg	1 mg	7 - 10 business days*	48.00€
TGM-T11234-5mg	5 mg	7 - 10 business days*	114.00€
TGM-T11234-1mL	1 ml	7 - 10 business days*	133.00€
TGM-T11234-10mg	10 mg	7 - 10 business days*	187.00€
TGM-T11234-25mg	25 mg	7 - 10 business days*	430.00€

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Description: ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 µM. ESI-08... more

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Product information "ESI-08"

Description: ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 µM. ESI-08 selectively blocks cAMP-induced EPAC activation but not cAMP-mediated PKA activation. Target: cAMP. Smiles: Cc1ccc(C)c(CSc2nc(C3CCCCC3)c(C#N)c(=O)[nH]2)c1. References: Chen H, et al. 5-Cyano-6-oxo-1,6-dihydro-pyrimidines as potent antagonists targeting exchange proteins directly activated by cAMP. Bioorg Med Chem Lett. 2012 Jun 15,22(12):4038-43.

Supplier:	TargetMol
Supplier-Nr:	T11234

Properties

MW:	353.48 D
Formula:	C20H23N3OS

Database Information

CAS :

301177-43-5| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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