ESI-05

Item number	Size	Delivery time	Price
TGM-T15247-2mg	2 mg	7 - 10 business days*	34.00€
TGM-T15247-5mg	5 mg	7 - 10 business days*	52.00€
TGM-T15247-1mL	1 ml	7 - 10 business days*	58.00€
TGM-T15247-10mg	10 mg	7 - 10 business days*	93.00€
TGM-T15247-25mg	25 mg	7 - 10 business days*	167.00€
TGM-T15247-50mg	50 mg	7 - 10 business days*	283.00€
TGM-T15247-100mg	100 mg	7 - 10 business days*	485.00€

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Description: ESI-05 (NSC-116966) is a specific EPAC2 (exchange protein directly activated by cAMP... more

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Product information "ESI-05"

Description: ESI-05 (NSC-116966) is a specific EPAC2 (exchange protein directly activated by cAMP 2) antagonist (IC50: 0.4 µM). ESI-05 inhibits cAMP-mediated activation of EPAC2, as well as EAPC2, mediated Rap1 activation. Target: cAMP. Smiles: Cc1ccc(cc1)S(=O)(=O)c1c(C)cc(C)cc1C. References: Tsalkova T, et al. Isoform-specific antagonists of exchange proteins directly activated by cAMP. Proc Natl Acad Sci U S A. 2012 Nov 6,109(45):18613-8.

Keywords:	NSC 116966
Supplier:	TargetMol
Supplier-Nr:	T15247

Properties

Application:	Rap guanine nucleotide exchange factor 4 (Epac2) inhibitor
MW:	274.38 D
Formula:	C16H18O2S

Database Information

CAS :	5184-64-5\| Matching products
KEGG ID :	K04351 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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