Encaleret

Item number	Size	Manual	Delivery time	Price
Cay45051-1	1 mg	-	6 - 10 business days*	169.00€
Cay45051-5	5 mg	-	6 - 10 business days*	506.00€
Cay45051-10	10 mg	-	6 - 10 business days*	842.00€

If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk

A CaSR antagonist (IC50 = 0.012 µM in a reporter assay using PC12h cells), increases plasma... more

Close menu

Product information "Encaleret"

A CaSR antagonist (IC50 = 0.012 µM in a reporter assay using PC12h cells), increases plasma levels of parathyroid hormone, prevents renal calcification, and increases bone mineral density in an ADH model using CaSR knock-in mice. SMILES: FC(C=C1CC(C)(C)NC[C@@H](O)CO[C@@H](C(C=CC=C2)=C2C3=CC(C)=C(C(O)=O)C=C3)C)=C(C=C1)Cl. InChi Code: InChI=1S/C29H33ClFNO4/c1-18-13-21(10-11-23(18)28(34)35)25-8-6-5-7-24(25)19(2)36-17-22(33)16-32-29(3,4)15-20-9-12-26(30)27(31)14-20/h5-14,19,22,32-33H,15-17H2,1-4H3,(H,34,35)/t19-,22-/m1/s1. InChi Key: UNFHDRVFEQPUEL-DENIHFKCSA-N

Keywords:	CLTX-305, JTT-305, MK-5442, 2'-[(1R)-1-[(2R)-3-[[2-(4-chloro-3-fluorophenyl)-1,1-dimethylethyl]amino]-2-hydroxypropoxy]ethyl]-3-methyl-[1,1'-biphenyl]-4-carboxylic acid
Supplier:	Cayman Chemical
Supplier-Nr:	45051

Properties

Application:	Osteoporosis agent, calcium-sensing receptor (CaSR) antagonist
MW:	514.03 D
Formula:	C29H33ClFNO4
Purity:	>95%
Format:	Solid

Database Information

CAS :	787583-71-5\| Matching products
KEGG ID :	K04612 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: -20°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

Information about the product reference will follow. more

Close menu

View product citations for antibody 45051 on CiteAb

You will get a certificate here

Go back

Read, write and discuss reviews... more

Close menu

Customer review for "Encaleret"

Write a review