Dexloxiglumide
| Item number | Size | Datasheet | Manual | SDS | Delivery time | Quantity | Price |
|---|---|---|---|---|---|---|---|
| Cay34759-10 | 10 mg | - |
6 - 10 business days* |
44.00€
|
|||
| Cay34759-25 | 25 mg | - |
6 - 10 business days* |
100.00€
|
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Dexloxiglumide is a cholecystokinin (CCK) receptor antagonist and is the single (R) isomer of... more
Product information "Dexloxiglumide"
Dexloxiglumide is a cholecystokinin (CCK) receptor antagonist and is the single (R) isomer of loxiglumide (Cay-25534). It selectively binds to the CCK1 receptor over CCK2 in CHO cells expressing the rat receptors (Kis = 0.0234 and 5.88 µM, respectively). Dexloxiglumide (20 µmol/kg) inhibits guinea pig gallbladder contractions induced by the CCK agonist CCK octapeptide (sulfated) (CCK-8S, Cay-23371). It reduces CCK-8-induced gastric emptying in rats (ID50 = 1.14 mg/kg).Formal Name: (4R)-4-[(3,4-dichlorobenzoyl)amino]-5-[(3-methoxypropyl)pentylamino]-5-oxo-pentanoic acid. CAS Number: 119817-90-2. Molecular Formula: C21H30Cl2N2O5. Formula Weight: 461.4. Purity: >98%. Formulation: (Request formulation change), A solid. Solubility: DMSO: 50 mg/ml, sonicated. SMILES: CCCCCN(CCCOC)C([C@@H](CCC(O)=O)NC(C1=CC(Cl)=C(C=C1)Cl)=O)=O. InChi Code: InChI=1S/C21H30Cl2N2O5/c1-3-4-5-11-25(12-6-13-30-2)21(29)18(9-10-19(26)27)24-20(28)15-7-8-16(22)17(23)14-15/h7-8,14,18H,3-6,9-13H2,1-2H3,(H,24,28)(H,26,27)/t18-/m1/s1. InChi Key: QNQZBKQEIFTHFZ-GOSISDBHSA-N.
| Keywords: | (4R)-4-[(3,4-dichlorobenzoyl)amino]-5-[(3-methoxypropyl)pentylamino]-5-oxo-pentanoic acid |
| Supplier: | Cayman Chemical |
| Supplier-Nr: | 34759 |
Properties
| Application: | CCK1 receptor antagonist |
| MW: | 461.4 D |
| Formula: | C21H30Cl2N2O5 |
| Purity: | >98% |
| Format: | Solid |
Database Information
| CAS : | 119817-90-2| Matching products |
| KEGG ID : | K04194 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +20°C (International: -20°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302, H315, H319, H335 |
| P Phrases: | P261, P264, P270, P271, P280, P312, P321, P330, P301+P310, P302+P352, P304+P340, P305+P351+P338, P332+P313, P337+P313, P362+P364, P405, P403+P233, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
Information about the product reference will follow.
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