CCG215022

Item number	Size	Delivery time	Price
TGM-T3498-1mg	1 mg	7 - 10 business days*	97.00€
TGM-T3498-2mg	2 mg	7 - 10 business days*	142.00€
TGM-T3498-5mg	5 mg	7 - 10 business days*	245.00€
TGM-T3498-1mL	1 ml	7 - 10 business days*	271.00€
TGM-T3498-10mg	10 mg	7 - 10 business days*	395.00€
TGM-T3498-25mg	25 mg	7 - 10 business days*	660.00€
TGM-T3498-50mg	50 mg	7 - 10 business days*	944.00€
TGM-T3498-100mg	100 mg	7 - 10 business days*	1,281.00€
TGM-T3498-500mg	500 mg	7 - 10 business days*	2,573.00€

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Description: CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of... more

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Product information "CCG215022"

Description: CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 µM for GRK2, 0.38±0.06 µM for GRK5, and 3.9±1 µM for GRK1. Target: PKA, GRK. Smiles: CC1=C(C(NC(=O)N1)c1ccc(F)c(c1)C(=O)NCc1ccccn1)C(=O)Nc1ccc2[nH]ncc2c1. References: Homan KT, et al. Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally DesignedInhibitor. J Biol Chem. 2015 Aug 21,290(34):20649-59.

Supplier:	TargetMol
Supplier-Nr:	T3498

Properties

Application:	GRK inhibitor
MW:	499.5 D
Formula:	C26H22FN7O3

Database Information

CAS :	1813527-81-9\| Matching products
KEGG ID :	K00909 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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